BDBM86751 CHEMBL14935::LY 293558::LY-293558

SMILES: OC(=O)[C@@H]1C[C@H]2C[C@@H](CCc3nnn[nH]3)CC[C@H]2CN1

InChI Key: InChIKey=ZXFRFPSZAKNPQQ-UHFFFAOYSA-N

Data: 21 KI  1 IC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 22 hits for monomerid = 86751   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Glutamate receptor ionotropic, kainate 1 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	500	n/a	n/a	n/a	n/a	n/a	n/a
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Glutamate receptor 2 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		2.21E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Glutamate receptor 2 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		3.20E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Glutamate receptor 2 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		3.20E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Glutamate receptor 2 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		3.20E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Glutamate receptor ionotropic, kainate 1 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		4.16E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Glutamate receptor ionotropic, kainate 5 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		4.20E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 1 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		4.20E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Glutamate receptor 1 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		9.20E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Glutamate receptor 1 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		9.20E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Glutamate receptor 4 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 2 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 3 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Glutamate receptor 3 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		3.20E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Glutamate receptor 3 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		3.20E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Glutamate receptor 4 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Glutamate receptor 4 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		5.05E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 2 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 3 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 2 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 2 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 2 (Human)	BDBM86751 (CHEMBL14935 | LY-293558 | LY 293558) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair