BDBM87558 US10245267, Example 739::US10709712, Example 739::US9694016, 739
SMILES: C[C@H](O)CNc1nc(cc(n1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C)N1CCOCC1
InChI Key: InChIKey=IWHDNPFVBLBMGN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 87558 Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kcal/mole | IC50
nM | Kd
nM | EC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Serine/threonine-protein kinase B-raf [V600E]
(Human) | BDBM87558
(US9694016, 739 | US10245267, Example 739 | US10709...) | GoogleScholar
| UniChem
| | n/a | n/a | 4.10 | n/a | n/a | n/a | n/a | 7.5 | 25 |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
RAF proto-oncogene serine/threonine-protein kinase [Y340E,Y341E]
(Human) | BDBM87558
(US9694016, 739 | US10245267, Example 739 | US10709...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | 7.5 | 25 |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Serine/threonine-protein kinase B-raf [V600E]
(Human) | BDBM87558
(US9694016, 739 | US10245267, Example 739 | US10709...) | GoogleScholar
| UniChem
| | n/a | n/a | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
RAF proto-oncogene serine/threonine-protein kinase
(Human) | BDBM87558
(US9694016, 739 | US10245267, Example 739 | US10709...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Serine/threonine-protein kinase B-raf [V600E]
(Human) | BDBM87558
(US9694016, 739 | US10245267, Example 739 | US10709...) | GoogleScholar
| UniChem
| | n/a | n/a | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
RAF proto-oncogene serine/threonine-protein kinase
(Human) | BDBM87558
(US9694016, 739 | US10245267, Example 739 | US10709...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
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