BDBM8970 CHEMBL51197::N-[7-(1,2,3,4-tetrahydroacridin-9-ylsulfanyl)heptyl]-1,2,3,4-tetrahydroacridin-9-amine::Tacrine Dimer 4f::tacrine heterobivalent compound 3e
SMILES C(CCCNc1c2CCCCc2nc2ccccc12)CCCSc1c2CCCCc2nc2ccccc12
InChI Key InChIKey=QRIQNQYNWBQHLY-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 8970
Affinity DataKi: 35nM ΔG°: -10.2kcal/molepH: 8.0 T: 2°CAssay Description:Inhibition of enzyme activity was measured over a substrate concentration range of 0.01-30 mM and at least six inhibitor concentrations to determine ...More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of Equine ButyrylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of enzyme activity was measured over a substrate concentration range of 0.01-30 mM and at least six inhibitor concentrations to determine ...More data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Inhibition of fetal Bovine serum AChEMore data for this Ligand-Target Pair
Affinity DataKi: 340nM ΔG°: -8.82kcal/molepH: 8.0 T: 2°CAssay Description:Inhibition of enzyme activity was measured over a substrate concentration range of 0.01-30 mM and at least six inhibitor concentrations to determine ...More data for this Ligand-Target Pair
Affinity DataKi: 340nM ΔG°: -8.82kcal/molepH: 8.0 T: 2°CAssay Description:Inhibition of enzyme activity was measured over a substrate concentration range of 0.01-30 mM and at least six inhibitor concentrations to determine ...More data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of fetal bovine serum AChE using acetylthiocholine iodide as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrateMore data for this Ligand-Target Pair