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Found 35 Enz. Inhib. hit(s) with Target = 'Interleukin-21'
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649500(US11891386, Compound ARI-120)
Affinity DataIC50:  0.300nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649497(US11891386, Compound ARI-083)
Affinity DataIC50:  0.300nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649499(US11891386, Compound ARI-118)
Affinity DataIC50:  0.800nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649495(US11891386, Compound ARI-056)
Affinity DataIC50:  4.90nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649503(US11891386, Compound ARI-148)
Affinity DataIC50:  5.90nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649487(US11891386, Compound ARI-067)
Affinity DataIC50:  6.30nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649498(US11891386, Compound ARI-090)
Affinity DataIC50:  8.40nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649489(US11891386, Compound ARI-140)
Affinity DataIC50:  8.60nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649505(US11891386, Compound ARI-049)
Affinity DataIC50:  10.1nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649502(US11891386, Compound ARI-146)
Affinity DataIC50:  13.4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649506(US11891386, Compound ARI-065)
Affinity DataIC50:  14nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649491(US11891386, Compound ARI-143)
Affinity DataIC50:  18.8nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649488(US11891386, Compound ARI-087)
Affinity DataIC50:  25.4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649492(US11891386, Compound ARI-149)
Affinity DataIC50:  30.3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM50506039(CHEMBL1324296 | US11891386, Compound 002)
Affinity DataIC50:  31.8nMMore data for this Ligand-Target Pair
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM50506039(CHEMBL1324296 | US11891386, Compound 002)
Affinity DataIC50:  38.2nMMore data for this Ligand-Target Pair
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649493(US11891386, Compound ARI-030)
Affinity DataIC50:  40nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649494(US11891386, Compound ARI-031)
Affinity DataIC50:  42.6nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649501(US11891386, Compound ARI-145)
Affinity DataIC50:  46.9nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649485(US11891386, Compound ARI-066)
Affinity DataIC50:  48.6nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649482(US11891386, Compound ARI-055)
Affinity DataIC50:  73.6nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649496(US11891386, Compound ARI-060)
Affinity DataIC50:  110nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM649490(US11891386, Compound ARI-142)
Affinity DataIC50:  209nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM50605060(CHEMBL5198290 | US11891386, Compound 004)
Affinity DataIC50:  231nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM247034(1-((1-(methylsulfonyl)piperidin-4-yl)methyl)-5-(1H...)
Affinity DataIC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM247010(1-((1-(phenylsulfonyl)piperidin-4-yl)methyl)-5-(1H...)
Affinity DataIC50: <1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM247033(US9701663, 48 | rac.-trans-1-((-5-methyl-1-(phenyl...)
Affinity DataIC50: <1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM247023(US9701663, 6)
Affinity DataIC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM247026(US9701663, 7)
Affinity DataIC50: <1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM247027(US9701663, 8)
Affinity DataIC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM247031(1-((1-(2-fluorophenylsulfonyl)piperidin-4-yl)methy...)
Affinity DataIC50: <1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM247029(1-((1-(4-chlorophenylsulfonyl)piperidin-4-yl)methy...)
Affinity DataIC50: <1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM247032(US9701663, 47 | rac.-cis-1-((-5-methyl-1-(phenylsu...)
Affinity DataIC50: <1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM247030(5-(1H-pyrazol-4-yl)-1-((1-(pyridin-3-ylsulfonyl)pi...)
Affinity DataIC50: <1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInterleukin-21(Homo sapiens (Human))TBA
LigandPNGBDBM247028(1-((5,5-dimethyl-1-(phenylsulfonyl)pyrrolidin-3-yl...)
Affinity DataIC50: <1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent