Affinity DataKi: 4.80nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Non-competitive inhibition of human recombinant LDHA assessed as inhibition constant using varying concentration of pyruvate as substrate preincubate...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 210nM ΔG°: -38.1kJ/mole IC50: 650nMpH: 7.5 T: 2°CAssay Description:An LDH enzymatic assay developed for high throughput format was used. The dehydrogenase reaction was run in the lactate to pyruvate direction and cou...More data for this Ligand-Target Pair
Affinity DataKi: 290nM ΔG°: -37.3kJ/mole IC50: 140nMpH: 7.5 T: 2°CAssay Description:An LDH enzymatic assay developed for high throughput format was used. The dehydrogenase reaction was run in the lactate to pyruvate direction and cou...More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Competitive inhibition of human LDH1 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 470nM ΔG°: -36.1kJ/mole IC50: 1.10E+3nMpH: 7.5 T: 2°CAssay Description:An LDH enzymatic assay developed for high throughput format was used. The dehydrogenase reaction was run in the lactate to pyruvate direction and cou...More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Non-competitive inhibition of human recombinant LDHB assessed as inhibition constant using varying concentration of pyruvate as substrate preincubate...More data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Competitive inhibition of human LDH1 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Non-competitive inhibition of human recombinant LDHA assessed as inhibition constant using varying concentration of pyruvate as substrate preincubate...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Competitive inhibition of human LDH1 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Mus musculus (Mouse))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition of mouse LDHB using sodium pyruvate as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Non-competitive inhibition of human recombinant LDHA assessed as inhibition constant using varying concentration of pyruvate as substrate preincubate...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Competitive inhibition of human LDH1 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Mixed inhibition of human recombinant LDHA assessed as inhibition constant using varying concentration of pyruvate as substrate preincubated for 10 m...More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Inhibition of human LDHA using sodium pyruvate as substrateMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Mixed inhibition of human recombinant LDHB assessed as inhibition constant using varying concentration of pyruvate as substrate preincubated for 10 m...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine
Curated by ChEMBL
University Of New Mexico School Of Medicine
Curated by ChEMBL
Affinity DataKi: 4.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nMAssay Description:Competitive inhibition of human LDH-A using pyruvate as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair