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Found 8490 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A'
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400125(CHEMBL2178426)
Affinity DataKi:  0.00500nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400133(CHEMBL2178987)
Affinity DataKi:  0.00500nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400112(CHEMBL2178439)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400111(CHEMBL2178440)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400110(CHEMBL2178441)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400121(CHEMBL2178430)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400123(CHEMBL2178428)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400129(CHEMBL2178991)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400103(CHEMBL2178985)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400105(CHEMBL2178983)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400118(CHEMBL2178433)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400107(CHEMBL2178981)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400115(CHEMBL2178436)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400109(CHEMBL2178442)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400114(CHEMBL2178437)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400131(CHEMBL2178989)
Affinity DataKi:  0.00600nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400113(CHEMBL2178438)
Affinity DataKi:  0.00700nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400128(CHEMBL2178992)
Affinity DataKi:  0.00700nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400127(CHEMBL2178993)
Affinity DataKi:  0.00700nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400124(CHEMBL2178427)
Affinity DataKi:  0.00700nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400119(CHEMBL2178432)
Affinity DataKi:  0.00700nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400120(CHEMBL2178431)
Affinity DataKi:  0.00700nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400117(CHEMBL2178434)
Affinity DataKi:  0.00700nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400116(CHEMBL2178435)
Affinity DataKi:  0.00700nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400106(CHEMBL2178982)
Affinity DataKi:  0.00800nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400108(CHEMBL2178980)
Affinity DataKi:  0.00900nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400122(CHEMBL2178429)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400126(CHEMBL2178425)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400104(CHEMBL2178984)
Affinity DataKi:  0.0110nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400134(CHEMBL2178986)
Affinity DataKi:  0.0110nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400130(CHEMBL2178990)
Affinity DataKi:  0.0110nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50400132(CHEMBL2178988)
Affinity DataKi:  0.0120nMAssay Description:Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universitat AutòNoma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50087809(CHEMBL298006 | Methyl-(1-methyl-1H-indol-2-ylmethy...)
Affinity DataKi:  0.300nMAssay Description:Inhibitory activity against Monoamine oxidase AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50232429(CHEMBL4104691)
Affinity DataKi:  0.480nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50361606(CHEMBL1939851)
Affinity DataKi:  0.600nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universitat AutòNoma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50087796((5-Methoxy-1-methyl-1H-indol-2-ylmethyl)-prop-2-yn...)
Affinity DataKi:  0.800nMAssay Description:Inhibitory activity against Monoamine oxidase AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50361609(CHEMBL1939853)
Affinity DataKi:  0.800nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A/B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179395(CHEMBL14640)
Affinity DataKi:  0.891nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A/B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179395(CHEMBL14640)
Affinity DataKi:  0.891nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50273531(CHEMBL460599 | N-Methyl,N-(3-phenylpropyl)-1H-indo...)
Affinity DataKi:  0.920nMAssay Description:Inhibition of bovine brain mitochondrial MAO-A by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50557361(CHEMBL4761363)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50557339(CHEMBL4748517)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50557368(CHEMBL4762228)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50557366(CHEMBL4787184)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50557363(CHEMBL4757953)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50273595(CHEMBL462097 | N-(1H-Indol-2-ylmethyl)-N-methyl-N-...)
Affinity DataKi:  1nMAssay Description:Inhibition of bovine brain mitochondrial MAO-A by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50361607(CHEMBL1938411)
Affinity DataKi:  1nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Ntz Lab

Curated by ChEMBL
LigandPNGBDBM50557360(CHEMBL4787516)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50475875(CHEMBL212501)
Affinity DataKi:  1nMAssay Description:Inhibition of bovine brain mitochondrial MAOAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universitat AutòNoma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50087791(But-2-ynyl-(5-methoxy-1-methyl-1H-indol-2-ylmethyl...)
Affinity DataKi:  1.40nMAssay Description:Inhibitory activity against Monoamine oxidase AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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