4MP2: crystal structure of pyruvate dehydrogenase kinase isoform 2 in complex with inhibitor pa1 (10.1074/JBC.M113.533885 )
4MP7: crystal structure of pyruvate dehydrogenase kinase isoform 2 in complex with inhibitor pa7 (10.1074/JBC.M113.533885 )
4MPC: crystal structure of pyruvate dehydrogenase kinase isoform 2 in complex with inhibitor ps2 (10.1074/JBC.M113.533885 )
4MPE: crystal structure of pyruvate dehydrogenase kinase isoform 2 in complex with inhibitor ps8 (10.1074/JBC.M113.533885 )
4MPN: crystal structure of pyruvate dehydrogenase kinase isoform 2 in complex with inhibitor ps10 (10.1074/JBC.M113.533885 )
4V25: ver-246608, a novel pan-isoform atp competitive inhibitor of pyruvate dehydrogenase kinase, disrupts warburg metabolism and induces context- dependent cytostasis in cancer cells (10.18632/ONCOTARGET.2656 )
4V26: ver-246608, a novel pan-isoform atp competitive inhibitor of pyruvate dehydrogenase kinase, disrupts warburg metabolism and induces context- dependent cytostasis in cancer cells (10.18632/ONCOTARGET.2656 )
5M4K: application of off-rate screening in the identification of novel pan- isoform inhibitors of pyruvate dehydrogenase kinase (10.1021/ACS.JMEDCHEM.6B01478 )
5M4M: application of off-rate screening in the identification of novel pan- isoform inhibitors of pyruvate dehydrogenase kinase (10.1021/ACS.JMEDCHEM.6B01478 )
5M4N: application of off-rate screening in the identification of novel pan- isoform inhibitors of pyruvate dehydrogenase kinase (10.1021/ACS.JMEDCHEM.6B01478 )
5M4P: application of off-rate screening in the identification of novel pan- isoform inhibitors of pyruvate dehydrogenase kinase (10.1021/ACS.JMEDCHEM.6B01478 )