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Found 219 with Last Name = 'amatruda' and Initial = 'j'
TargetProtein Wnt-2(Mus musculus (Mouse))
University Of Texas Southwestern Medical Center

LigandPNGBDBM36414(CID15993586 | trans-N-Benzyl-4-((1-((2-cyanophenyl...)
Affinity DataIC50:  25nMpH: 7.4 T: 2°CAssay Description:Inhibition assay of Wnt response treated with exogenously supplied of Wnt protein ('exogenous Wnt' test)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Wnt-2(Mus musculus (Mouse))
University Of Texas Southwestern Medical Center

LigandPNGBDBM36412(CID25093486 | N-(4-Methylquinolin-8-yl)-4-(endo-4-...)
Affinity DataIC50:  27nMpH: 7.4 T: 2°CAssay Description:Inhibition assay of Wnt response treated with exogenously supplied of Wnt protein ('exogenous Wnt' test)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Wnt-2(Mus musculus (Mouse))
University Of Texas Southwestern Medical Center

LigandPNGBDBM36413(CID15995771 | trans-N-Benzyl-4-((1-((6-methyl-4-ox...)
Affinity DataIC50:  40nMpH: 7.4 T: 2°CAssay Description:Inhibition assay of Wnt response treated with exogenously supplied of Wnt protein ('exogenous Wnt' test)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Wnt-2(Mus musculus (Mouse))
University Of Texas Southwestern Medical Center

LigandPNGBDBM50294835(4-((1S,2S,6R,7R)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*...)
Affinity DataIC50:  58nMpH: 7.4 T: 2°CAssay Description:Inhibition assay of Wnt response treated with exogenously supplied of Wnt protein ('exogenous Wnt' test)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216934(2-((S)-5-(2-(2-(3-fluorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216935(2-(3,3-dimethyl-5-(2-(5-methyl-2-phenyloxazol-4-yl...)
Affinity DataEC50:  6.48E+3nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216936((S)-2-(5-(2-(2-(4-ethylphenyl)-1,4-dimethyl-1H-imi...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216937((S)-2-(5-(2-(2-(4-chlorophenyl)-5-methylthiazol-4-...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216939(CHEMBL246207 | {(S)-5-[2-(2-biphenyl-4-yl-5-methyl...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216943(2-((S)-5-(2-(2-(3-fluorophenyl)-5-methylthiazol-4-...)
Affinity DataEC50:  47nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216940(2-((S)-5-(2-(2-(benzo[d][1,3]dioxol-5-yl)-5-methyl...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216941((S)-2-(5-(2-(2-(4-isopropylphenyl)-5-methyloxazol-...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216938((S)-2-(5-(2-(2-(4-methoxyphenyl)-1,5-dimethyl-1H-i...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216944((S)-2-(6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-...)
Affinity DataEC50:  3.14E+3nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50176631(2-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2,3-...)
Affinity DataEC50:  590nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216947((S)-2-(5-(2-(5-ethyl-2-p-tolyloxazol-4-yl)ethoxy)-...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216945((S)-2-(5-(2-(2-(4-chlorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216946((S)-2-(5-(2-(5-ethyl-2-(4-ethylphenyl)oxazol-4-yl)...)
Affinity DataEC50:  2.53E+3nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216938((S)-2-(5-(2-(2-(4-methoxyphenyl)-1,5-dimethyl-1H-i...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216948((S)-2-(5-(2-(2-(4-ethylphenyl)-5-methyloxazol-4-yl...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216949(2-((S)-5-(2-(5-methyl-2-m-tolyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  64nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216951((S)-2-(5-(2-(2-(4-fluorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216943(2-((S)-5-(2-(2-(3-fluorophenyl)-5-methylthiazol-4-...)
Affinity DataEC50:  6.53E+3nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216950(2-((S)-5-(2-(2-(3-cyanophenyl)-5-methyloxazol-4-yl...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216953(2-((S)-5-(2-(5-methyl-2-m-tolylthiazol-4-yl)ethoxy...)
Affinity DataEC50:  6.79E+3nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216954((S)-2-(5-(2-(2-phenyl-5-propyloxazol-4-yl)ethoxy)-...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50176631(2-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2,3-...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216957((S)-2-(5-(2-(2-(4-tert-butylphenyl)-5-methyloxazol...)
Affinity DataEC50:  546nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216955((S)-2-(5-(2-(5-phenethyl-2-phenyloxazol-4-yl)ethox...)
Affinity DataEC50:  607nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50176673(2-methoxy-2-(5-(2-(5-methyl-2-phenyloxazol-4-yl)et...)
Affinity DataEC50:  4.40E+3nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216956((S)-2-(5-(2-(5-methyl-2-p-tolyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216958((S)-2-(5-(2-(1,5-dimethyl-2-phenyl-1H-imidazol-4-y...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216933(2-((S)-5-(2-(5-methyl-2-(3-(trifluoromethyl)phenyl...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216934(2-((S)-5-(2-(2-(3-fluorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  1.69E+3nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216959((S)-2-(5-(2-(1,4-dimethyl-2-phenyl-1H-imidazol-5-y...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216960((S)-2-(5-(2-(5-methyl-2-p-tolylthiazol-4-yl)ethoxy...)
Affinity DataEC50:  594nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216960((S)-2-(5-(2-(5-methyl-2-p-tolylthiazol-4-yl)ethoxy...)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216961((S)-2-(5-(2-(2-(4-methoxyphenyl)-1,4-dimethyl-1H-i...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216932(2-((S)-5-(2-(2-(3-chlorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  1.57E+3nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216957((S)-2-(5-(2-(2-(4-tert-butylphenyl)-5-methyloxazol...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216962((S)-2-(5-(2-(2-(4-isopropylphenyl)-5-methylthiazol...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216965((S)-2-(5-(2-(5-methyl-2-(4-(trifluoromethoxy)pheny...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216932(2-((S)-5-(2-(2-(3-chlorophenyl)-5-methyloxazol-4-y...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216967(CHEMBL428929 | {(S)-5-[2-(2-biphenyl-4-yl-1,5-dime...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216964((S)-2-(5-(2-(2-(4-ethoxyphenyl)-5-methylthiazol-4-...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216963((S)-2-(5-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216970(2-(6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2,3-...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216940(2-((S)-5-(2-(2-(benzo[d][1,3]dioxol-5-yl)-5-methyl...)
Affinity DataEC50:  1.21E+3nMAssay Description:Agonist activity at PPARalpha by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216969(2-(2-methyl-5-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataEC50:  883nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50216936((S)-2-(5-(2-(2-(4-ethylphenyl)-1,4-dimethyl-1H-imi...)
Affinity DataEC50:  31nMAssay Description:Agonist activity at GST-tagged human PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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