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Found 94 with Last Name = 'amer' and Initial = 'mf'
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180584(CHEMBL3814496)
Affinity DataIC50:  42nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180583(CHEMBL3815109)
Affinity DataIC50:  90nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180582(CHEMBL3814988)
Affinity DataIC50:  90nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180520(CHEMBL3814838)
Affinity DataIC50:  120nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180584(CHEMBL3814496)
Affinity DataIC50:  150nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180584(CHEMBL3814496)
Affinity DataIC50:  210nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180580(CHEMBL3814911)
Affinity DataIC50:  240nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180580(CHEMBL3814911)
Affinity DataIC50:  250nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180520(CHEMBL3814838)
Affinity DataIC50:  270nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180583(CHEMBL3815109)
Affinity DataIC50:  280nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50338672(CHEMBL1209027 | Salaprinol)
Affinity DataIC50:  290nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180586(CHEMBL1182462)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180582(CHEMBL3814988)
Affinity DataIC50:  340nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180588(CHEMBL3814747)
Affinity DataIC50:  390nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50242271((2R,3R,4R,5S)-1-(2-hydroxyethyl)-2-(hydroxymethyl)...)
Affinity DataIC50:  430nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180588(CHEMBL3814747)
Affinity DataIC50:  460nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180583(CHEMBL3815109)
Affinity DataIC50:  470nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180579(CHEMBL3814555)
Affinity DataIC50:  470nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180579(CHEMBL3814555)
Affinity DataIC50:  500nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180580(CHEMBL3814911)
Affinity DataIC50:  640nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180582(CHEMBL3814988)
Affinity DataIC50:  690nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataIC50:  750nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataIC50:  750nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180581(CHEMBL3814264)
Affinity DataIC50:  950nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180520(CHEMBL3814838)
Affinity DataIC50:  960nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180581(CHEMBL3814264)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180585(CHEMBL239249)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180581(CHEMBL3814264)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180586(CHEMBL1182462)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180579(CHEMBL3814555)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180585(CHEMBL239249)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50394353(CHEMBL2159763)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5R,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5R,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180588(CHEMBL3814747)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50338672(CHEMBL1209027 | Salaprinol)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338672(CHEMBL1209027 | Salaprinol)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50242271((2R,3R,4R,5S)-1-(2-hydroxyethyl)-2-(hydroxymethyl)...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50242271((2R,3R,4R,5S)-1-(2-hydroxyethyl)-2-(hydroxymethyl)...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of rat small intestinal isomaltase using isomaltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50180585(CHEMBL239249)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of human small intestine microsomal maltase using maltose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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