TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Bioprojet-Biotech
Curated by ChEMBL
Bioprojet-Biotech
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from human sigma1 receptor measured after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Bioprojet-Biotech
Curated by ChEMBL
Bioprojet-Biotech
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from human sigma1 receptor measured after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Bioprojet-Biotech
Curated by ChEMBL
Bioprojet-Biotech
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-(+)-pentazocine from human sigma1 receptor measured after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Bioprojet-Biotech
Curated by ChEMBL
Bioprojet-Biotech
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]-(+)-pentazocine from human sigma1 receptor measured after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Bioprojet-Biotech
Curated by ChEMBL
Bioprojet-Biotech
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D4.4 receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D4.4 receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]spiperone from recombinant human D4 receptor stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D4.4 receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Bioprojet-Biotech
Curated by ChEMBL
Bioprojet-Biotech
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-(+)-pentazocine from human sigma1 receptor measured after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 144nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D4.4 receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D4.4 receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Bioprojet-Biotech
Curated by ChEMBL
Bioprojet-Biotech
Curated by ChEMBL
Affinity DataKi: 4.60E+3nMAssay Description:Displacement of [3H]dofetilide from recombinant human ERG stably expressed in HEK293 cell membranes measured after 60 mins by scintillation counting ...More data for this Ligand-Target Pair
Affinity DataKi: 6.30E+3nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D2S receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor measured after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Chemveda Life Sciences India
Curated by ChEMBL
Chemveda Life Sciences India
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human CLK1 (130 to end residues) using ERMRPRKRQGSVRRRV as substrate incubated for 40 mins in presence of [gamma33P-ATP] by...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Chemveda Life Sciences India
Curated by ChEMBL
Chemveda Life Sciences India
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human CLK1 (130 to end residues) using ERMRPRKRQGSVRRRV as substrate incubated for 40 mins in presence of [gamma33P-ATP] by...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))
Chemveda Life Sciences India
Curated by ChEMBL
Chemveda Life Sciences India
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human CLK4 (128 to end residues) using YRRAAVPPSPSLSRHSSPHQS(p)EDEEE as substrate incubated for 40 mins in presence of [gam...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Chemveda Life Sciences India
Curated by ChEMBL
Chemveda Life Sciences India
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human CLK2 (138 to end residues) using YRRAAVPPSPSLSRHSSPHQS(p)EDEEE as substrate incubated for 40 mins in presence of [gam...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Chemveda Life Sciences India
Curated by ChEMBL
Chemveda Life Sciences India
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of rat DYRK1A (1 to 499 residues) assessed as residual activity by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK3(Homo sapiens (Human))
Chemveda Life Sciences India
Curated by ChEMBL
Chemveda Life Sciences India
Curated by ChEMBL
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of recombinant human full length CLK3 using ERMRPRKRQGSVRRRV as substrate incubated for 40 mins in presence of [gamma33P-ATP] by scintilla...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Chemveda Life Sciences India
Curated by ChEMBL
Chemveda Life Sciences India
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of rat DYRK1A (1 to 499 residues) assessed as residual activity by ADP-Glo assayMore data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 3.49E+4nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 7.99E+4nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.01E+5nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.11E+5nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
Institute Of Chemical Technology
Curated by ChEMBL
Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 2.13E+5nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair