Compile Data Set for Download or QSAR
maximum 50k data
Found 50 with Last Name = 'araki' and Initial = 'm'
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054109(CHEMBL3319301)
Affinity DataIC50:  44nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054192(CHEMBL3319304)
Affinity DataIC50:  110nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054192(CHEMBL3319304)
Affinity DataIC50:  110nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054187(CHEMBL3319303)
Affinity DataIC50:  111nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054187(CHEMBL3319303)
Affinity DataIC50:  111nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054136(CHEMBL3319302)
Affinity DataIC50:  120nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50158866(CHEMBL3785355)
Affinity DataIC50:  132nMAssay Description:Inhibition of recombinant human LSD1 using H3K4me2 peptide as substrate measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054108(CHEMBL3356912)
Affinity DataIC50:  520nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50460073(CHEMBL4227224)
Affinity DataIC50:  622nMAssay Description:Inhibition of recombinant human LSD1 using H3K4me2 peptide as substrate measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50431886(CHEMBL1413473)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-(-)-2-phenylcyclopropylamine | (1R,2S)-2-p...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using (4S)-4,5-dihydro-2-(6-hydroxybenzothiazolyl)-4-thiazol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-(-)-2-phenylcyclopropylamine | (1R,2S)-2-p...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using (4S)-4,5-dihydro-2-(6-hydroxybenzothiazolyl)-4-thiazol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50009200(CHEMBL3238374)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093550(CHEMBL3585737)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of urokinase (unknown origin) using Pyr-Gly-Arg-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093544(CHEMBL3585744)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093552(CHEMBL3585735)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of urokinase (unknown origin) using Pyr-Gly-Arg-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093551(CHEMBL3585736)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50009171(CHEMBL3238362)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093553(CHEMBL3585734)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of urokinase (unknown origin) using Pyr-Gly-Arg-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093540(CHEMBL3585746)
Affinity DataIC50:  5.60E+4nMAssay Description:Inhibition of urokinase (unknown origin) using Pyr-Gly-Arg-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093541(CHEMBL3585745)
Affinity DataIC50:  7.40E+4nMAssay Description:Inhibition of urokinase (unknown origin) using Pyr-Gly-Arg-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-(-)-2-phenylcyclopropylamine | (1R,2S)-2-p...)
Affinity DataIC50:  8.07E+4nMAssay Description:Inhibition of recombinant human LSD1 using H3K4me2 peptide as substrate measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093542(CHEMBL3585742)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50158866(CHEMBL3785355)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using (4S)-4,5-dihydro-2-(6-hydroxybenzothiazolyl)-4-thiazol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50460073(CHEMBL4227224)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using (4S)-4,5-dihydro-2-(6-hydroxybenzothiazolyl)-4-thiazol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50158866(CHEMBL3785355)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using (4S)-4,5-dihydro-2-(6-hydroxybenzothiazolyl)-4-thiazol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine

Curated by ChEMBL
LigandPNGBDBM50460073(CHEMBL4227224)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using (4S)-4,5-dihydro-2-(6-hydroxybenzothiazolyl)-4-thiazol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093549(CHEMBL3585738)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093548(CHEMBL3585739)
Affinity DataIC50:  1.60E+5nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093541(CHEMBL3585745)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093540(CHEMBL3585746)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50009200(CHEMBL3238374)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093542(CHEMBL3585742)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093547(CHEMBL3585740)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093545(CHEMBL3585743)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093546(CHEMBL3585741)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50093543(CHEMBL3585747)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50009171(CHEMBL3238362)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of plasmin (unknown origin) using Boc-Val-Leu-Lys-MCA as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50203072(3-isothiocyanatoprop-1-ene | Allyl isothiocyanate ...)
Affinity DataEC50:  8.12E+3nMAssay Description:Agonist activity at TRPA1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50548720(CHEBI:42438 | CHEMBL1232595)
Affinity DataEC50:  8.28E+4nMAssay Description:Agonist activity at TRPA1 (unknown origin) by calcium imaging assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM36301(2-Chlorophenol (2-CP) | 2-chlorophenol)
Affinity DataEC50:  5.01E+5nMAssay Description:Agonist activity at TRPA1 (unknown origin) by calcium imaging assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50548721(CHEMBL3186900)
Affinity DataEC50:  1.01E+5nMAssay Description:Agonist activity at TRPA1 (unknown origin) by calcium imaging assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50548722(CHEMBL1490403)
Affinity DataEC50:  8.60E+4nMAssay Description:Agonist activity at TRPA1 (unknown origin) by calcium imaging assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50548725(3-Methylcatechol | CHEBI:18404 | CHEMBL1173328)
Affinity DataEC50:  2.83E+3nMAssay Description:Agonist activity at TRPA1 (unknown origin) by calcium imaging assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50548723(CHEBI:17254 | CHEMBL158766)
Affinity DataEC50:  1.17E+4nMAssay Description:Agonist activity at TRPA1 (unknown origin) by calcium imaging assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50094702(1H-indole | CHEMBL15844 | Indol | Indole, 7 | indo...)
Affinity DataEC50:  7.52E+4nMAssay Description:Agonist activity at TRPA1 (unknown origin) by calcium imaging assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50164168(1,3,4-Eugenol | 1-Hydroxy-2-methoxy-4-allylbenzene...)
Affinity DataEC50:  1.16E+5nMAssay Description:Agonist activity at TRPA1 (unknown origin) by calcium imaging assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50548724(CHEBI:50545 | CHEMBL193598)
Affinity DataEC50:  1.49E+5nMAssay Description:Agonist activity at TRPA1 (unknown origin) by calcium imaging assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50240432(1-hydroxy-5-methyl-2-isopropylbenzene | 2-isopropy...)
Affinity DataEC50:  8.69E+4nMAssay Description:Agonist activity at TRPA1 (unknown origin) by calcium imaging assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50483042(CHEMBL1276241)
Affinity DataEC50:  8.69E+3nMAssay Description:Agonist activity at TRPA1 (unknown origin) by calcium imaging assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed