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Found 43 with Last Name = 'azizeh' and Initial = 'by'
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(CHEMBL266481 | GLUCAGON | His-Ser-Gln-Gly-Thr-Phe-...)
Affinity DataIC50:  1.5nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051588(CHEMBL429362 | His-Ser-Gln-thr-Phe-Thr-Ser-Asp-Tyr...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(CHEMBL266481 | GLUCAGON | His-Ser-Gln-Gly-Thr-Phe-...)
Affinity DataIC50:  1.5nMAssay Description:Compound was tested for its ability to displace [I-125]-glucagon from the glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051586(CHEMBL413666 | [des-His1,Tyr5,Glu9,D-Tyr10]glucago...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50407844(CHEMBL2115191)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50454201(CHEMBL3037804)
Affinity DataIC50:  10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059352(CHEMBL442499 | [des-His1, Trp6, Glu9] glucagon-NH2)
Affinity DataIC50:  19nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50407842(CHEMBL2114176)
Affinity DataIC50:  34.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059358(CHEMBL267885 | [des-His1, Tyr6,Glu9] glucagon-NH2)
Affinity DataIC50:  40nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059362(CHEMBL268636 | [des-His1, des-Phe6, Glu9] glucagon...)
Affinity DataIC50:  48nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50284992(CHEMBL441209 | H-Ser-Gln-GlyThr-Thr-Ser-Glu-Tyr-Se...)
Affinity DataIC50:  48nMAssay Description:pA2 value towards glucagon receptor relative to glucagon was calculatedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059356(CHEMBL2369990 | [des-His1, Nle6, Glu9] glucagon-NH...)
Affinity DataIC50:  48nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059359(CHEMBL411289 | [des-His1, des-Gly4, Glu9] glucagon...)
Affinity DataIC50:  52nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051585(CHEMBL2369127 | [des-His1,Tyr5,Glu9,(2S,3R)-beta-M...)
Affinity DataIC50:  74nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059364(CHEMBL2369985 | [des-His1, D-Phe6, Glu9] glucagon-...)
Affinity DataIC50:  100nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059365(CHEMBL412352 | [des-Phe6, Glu9] glucagon-NH2)
Affinity DataIC50:  113nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059363(CHEMBL437095 | [des-His1,Ala6, Glu9] glucagon-NH2)
Affinity DataIC50:  126nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059360(CHEMBL429198 | [des-His1, des-Phe6] glucagon-NH2)
Affinity DataIC50:  128nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50032172((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)
Affinity DataIC50:  170nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50032172((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)
Affinity DataIC50:  180nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059361(CHEMBL439271 | [des-His1, des-Phe6] glucagon)
Affinity DataIC50:  200nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50407843(CHEMBL2114177)
Affinity DataIC50:  395nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059355(CHEMBL409611 | [des-Phe6] glucagon)
Affinity DataIC50:  500nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50407841(CHEMBL2115192)
Affinity DataIC50:  510nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059354(CHEMBL438574 | [des-Phe6] glucagon-NH2)
Affinity DataIC50:  512nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059351(CHEMBL427744 | [des-His1, des-Phe6, Glu9] glucagon...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059351(CHEMBL427744 | [des-His1, des-Phe6, Glu9] glucagon...)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059357(CHEMBL438218 | [des-His1, Asp6, Glu9] glucagon-NH2)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059357(CHEMBL438218 | [des-His1, Asp6, Glu9] glucagon-NH2)
Affinity DataKd:  501nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059361(CHEMBL439271 | [des-His1, des-Phe6] glucagon)
Affinity DataKd:  708nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059355(CHEMBL409611 | [des-Phe6] glucagon)
Affinity DataKd:  562nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059362(CHEMBL268636 | [des-His1, des-Phe6, Glu9] glucagon...)
Affinity DataKd:  6.31nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059358(CHEMBL267885 | [des-His1, Tyr6,Glu9] glucagon-NH2)
Affinity DataKd:  631nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059359(CHEMBL411289 | [des-His1, des-Gly4, Glu9] glucagon...)
Affinity DataKd:  891nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059363(CHEMBL437095 | [des-His1,Ala6, Glu9] glucagon-NH2)
Affinity DataKd:  398nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059352(CHEMBL442499 | [des-His1, Trp6, Glu9] glucagon-NH2)
Affinity DataKd:  562nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059351(CHEMBL427744 | [des-His1, des-Phe6, Glu9] glucagon...)
Affinity DataKd:  794nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059360(CHEMBL429198 | [des-His1, des-Phe6] glucagon-NH2)
Affinity DataKd:  562nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059354(CHEMBL438574 | [des-Phe6] glucagon-NH2)
Affinity DataKd:  501nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059365(CHEMBL412352 | [des-Phe6, Glu9] glucagon-NH2)
Affinity DataKd:  631nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059356(CHEMBL2369990 | [des-His1, Nle6, Glu9] glucagon-NH...)
Affinity DataKd:  501nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(CHEMBL266481 | GLUCAGON | His-Ser-Gln-Gly-Thr-Phe-...)
Affinity DataEC50:  8nMAssay Description:cAMP accumulation in rat hepatocytes in the presence rolipramMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 5(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051588(CHEMBL429362 | His-Ser-Gln-thr-Phe-Thr-Ser-Asp-Tyr...)
Affinity DataEC50:  8nMAssay Description:Ability of the Compound to activate Adenylate cyclase activity was measured by the conversion of [alpha-32P]ATP to 3'5'-cyclic AMPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed