Affinity DataIC50: 1.5nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Compound was tested for its ability to displace [I-125]-glucagon from the glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 34.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:pA2 value towards glucagon receptor relative to glucagon was calculatedMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 113nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 128nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 395nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 512nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataKd: 501nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataKd: 708nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataKd: 562nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataKd: 6.31nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataKd: 631nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataKd: 891nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataKd: 398nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataKd: 562nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataKd: 794nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataKd: 562nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataKd: 501nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataKd: 631nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataKd: 501nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:cAMP accumulation in rat hepatocytes in the presence rolipramMore data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:Ability of the Compound to activate Adenylate cyclase activity was measured by the conversion of [alpha-32P]ATP to 3'5'-cyclic AMPMore data for this Ligand-Target Pair