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Found 84 with Last Name = 'berlin' and Initial = 'kd'
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50335530((S)-3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-2,3-d...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50294211(3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-3-hydroxy...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50336512((R)-3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-2,3-d...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM18069(5-[(3,4,5-trimethoxyphenyl)methyl]pyrimidine-2,4-d...)
Affinity DataKi:  4.40nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM18070(5-[(2-cyclopropyl-7,8-dimethoxy-2H-chromen-5-yl)me...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM18070(5-[(2-cyclopropyl-7,8-dimethoxy-2H-chromen-5-yl)me...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50336514((S)-Iclaprim | CHEMBL1673303)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50336513((R)-Iclaprim | 5-[[(2R)-2-cyclopropyl-7,8-dimethox...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50335530((S)-3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-2,3-d...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50335530((S)-3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-2,3-d...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50294211(3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-3-hydroxy...)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50294211(3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-3-hydroxy...)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50336512((R)-3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-2,3-d...)
Affinity DataIC50:  11.5nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50336512((R)-3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-2,3-d...)
Affinity DataIC50:  11.5nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM18069(5-[(3,4,5-trimethoxyphenyl)methyl]pyrimidine-2,4-d...)
Affinity DataIC50:  14.4nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Bacillus anthracis)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM18050(2-[(4-{[(2,4-diaminopteridin-6-yl)methyl](methyl)a...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Bacillus anthracis DHFRMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Bacillus anthracis)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM18050(2-[(4-{[(2,4-diaminopteridin-6-yl)methyl](methyl)a...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Bacillus anthracis DHFRMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Bacillus anthracis)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50335531(1-propyl-2-acryloyl-1,2-dihydrophthalazine | CHEMB...)
Affinity DataIC50:  46nMAssay Description:Inhibition of Bacillus anthracis DHFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Bacillus anthracis)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50335530((S)-3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-2,3-d...)
Affinity DataIC50:  54nMAssay Description:Inhibition of Bacillus anthracis DHFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50298821((S)-5-(3-(2-methoxy-2',6'-dimethylbiphenyl-4-yl)bu...)
Affinity DataIC50:  61nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Staphylococcus aureus)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM25826(5-[(3R)-3-(3-methoxy-5-phenylphenyl)but-1-yn-1-yl]...)
Affinity DataIC50:  61nMAssay Description:Inhibition of Staphylococcus aureus wild type recombinant DHFR by MTS assayMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Bacillus anthracis)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50335532((E)-3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-2,3-d...)
Affinity DataIC50:  96nMAssay Description:Inhibition of Bacillus anthracis DHFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Bacillus anthracis)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50335533((E)-1-(1-butylphthalazin-2(1H)-yl)-3-(5-((2,4-diam...)
Affinity DataIC50:  170nMAssay Description:Inhibition of Bacillus anthracis DHFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Bacillus anthracis)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM18069(5-[(3,4,5-trimethoxyphenyl)methyl]pyrimidine-2,4-d...)
Affinity DataIC50:  7.70E+4nMAssay Description:Inhibition of Bacillus anthracis DHFRMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Bacillus anthracis)
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50095890(2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperaz...)
Affinity DataIC50:  1.02E+5nMAssay Description:Inhibition of Bacillus anthracis DHFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50335530((S)-3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-2,3-d...)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibition of human DHFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Oklahoma State University

Curated by ChEMBL
LigandPNGBDBM50294211(3-(5-((2,4-diaminopyrimidin-5-yl)methyl)-3-hydroxy...)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibition of human DHFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066900((2E,4E,6E)-7-(4,4-Dimethyl-thiochroman-6-yl)-3-met...)
Affinity DataEC50:  2.70E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066899((2E,4E,6E)-7-(4,4-Dimethyl-chroman-6-yl)-3-methyl-...)
Affinity DataEC50:  39nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066898(4-[(E)-2-(3,3-Dimethyl-2,3-dihydro-benzofuran-5-yl...)
Affinity DataEC50:  2.30E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066901((2E,4E,6E)-7-(3,3-Dimethyl-2,3-dihydro-benzo[b]thi...)
Affinity DataEC50:  8nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066898(4-[(E)-2-(3,3-Dimethyl-2,3-dihydro-benzofuran-5-yl...)
Affinity DataEC50:  320nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-beta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066902((2E,4E,6E)-7-(3,3-Dimethyl-2,3-dihydro-benzofuran-...)
Affinity DataEC50:  2.80E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066901((2E,4E,6E)-7-(3,3-Dimethyl-2,3-dihydro-benzo[b]thi...)
Affinity DataEC50:  2.60E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066903(4-[(E)-2-(3,3-Dimethyl-2,3-dihydro-benzofuran-5-yl...)
Affinity DataEC50:  400nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066900((2E,4E,6E)-7-(4,4-Dimethyl-thiochroman-6-yl)-3-met...)
Affinity DataEC50:  12nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066902((2E,4E,6E)-7-(3,3-Dimethyl-2,3-dihydro-benzofuran-...)
Affinity DataEC50:  230nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066902((2E,4E,6E)-7-(3,3-Dimethyl-2,3-dihydro-benzofuran-...)
Affinity DataEC50:  770nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-beta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066901((2E,4E,6E)-7-(3,3-Dimethyl-2,3-dihydro-benzo[b]thi...)
Affinity DataEC50:  1.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066902((2E,4E,6E)-7-(3,3-Dimethyl-2,3-dihydro-benzofuran-...)
Affinity DataEC50:  800nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066904(4-[(E)-2-(4,4-Dimethyl-chroman-6-yl)-propenyl]-ben...)
Affinity DataEC50:  140nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-beta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066904(4-[(E)-2-(4,4-Dimethyl-chroman-6-yl)-propenyl]-ben...)
Affinity DataEC50:  330nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066907(4-[(E)-2-(3,3-Dimethyl-2,3-dihydro-benzo[b]thiophe...)
Affinity DataEC50:  420nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066905(4-[(E)-2-(4,4-Dimethyl-chroman-6-yl)-propenyl]-ben...)
Affinity DataEC50:  1.10E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066906(4-[(E)-2-(4,4-Dimethyl-thiochroman-6-yl)-propenyl]...)
Affinity DataEC50:  620nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066898(4-[(E)-2-(3,3-Dimethyl-2,3-dihydro-benzofuran-5-yl...)
Affinity DataEC50:  460nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066904(4-[(E)-2-(4,4-Dimethyl-chroman-6-yl)-propenyl]-ben...)
Affinity DataEC50:  1.10E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066899((2E,4E,6E)-7-(4,4-Dimethyl-chroman-6-yl)-3-methyl-...)
Affinity DataEC50:  2.80E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066905(4-[(E)-2-(4,4-Dimethyl-chroman-6-yl)-propenyl]-ben...)
Affinity DataEC50:  200nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Oklahoma Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50066899((2E,4E,6E)-7-(4,4-Dimethyl-chroman-6-yl)-3-methyl-...)
Affinity DataEC50:  72nMAssay Description:Transcriptional activation in CV-1 cells expressing RAR-beta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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