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Found 205 with Last Name = 'bouloc' and Initial = 'n'
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467114(CHEMBL4285682)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467117(CHEMBL4288816)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467123(CHEMBL4288103)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467126(CHEMBL4286880)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467122(CHEMBL4279865)
Affinity DataIC50:  1nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467128(CHEMBL4286841)
Affinity DataIC50:  2nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318595(6-Bromo-7-[4-(5-methyl-isoxazol-3-ylmethyl)-pipera...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318575(2-{4-[6-Chloro-2-(4-morpholin-4-ylmethylphenyl)-3H...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318610(6-Bromo-7-[4-(5-methyl-isoxazol-3-ylmethyl)-pipera...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50182362(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318601(4-((4-(6-Bromo-2-(4-methoxyphenyl)-3H-imidazo[4,5-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318588(6-Bromo-2-(4-morpholin-4-ylmethyl-phenyl)-7-(4-pyr...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467127(CHEMBL4284547)
Affinity DataIC50:  6nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318590(4-(4-(6-Bromo-7-(4-(pyrimidin-5-ylmethyl)piperazin...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318602(4-(4-(6-Bromo-7-(4-(thiazol-4-ylmethyl)piperazin-1...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50168171(4-(2-(4-fluorophenyl)-5-(1-methylpiperidin-4-yl)-1...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467124(CHEMBL4283774)
Affinity DataIC50:  6nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318589(6-Bromo-2-(4-methoxyphenyl)-7-(4-(pyrimidin-5-ylme...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467116(CHEMBL4287934)
Affinity DataIC50:  9nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318587(6-Bromo-2-(4-methoxyphenyl)-7-(4-(pyridin-3-ylmeth...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318605((4-(6-Bromo-7-(4-((5-methylisoxazol-3-yl)methyl)pi...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318597(3-((4-(6-Chloro-2-(4-(4-methylpiperazin-1-yl)pheny...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318611(3-((4-(2-(4-((1H-Pyrazol-1-yl)methyl)phenyl)-6-chl...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318609(3-((4-(6-Bromo-2-(4-(piperazin-1-yl)phenyl)-3H-imi...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318603(3-((4-(6-Bromo-2-(4-(piperazin-1-ylmethyl)phenyl)-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318592(6-BROMO-7-[4-(4-CHLOROBENZYL)PIPERAZIN-1-YL]-2-[4-...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318604(1-(4-(6-Bromo-7-(4-((5-methylisoxazol-3-yl)methyl)...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318596(3-((4-(6-Bromo-2-(4-(4-methylpiperazin-1-yl)phenyl...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467121(CHEMBL4282026)
Affinity DataIC50:  15nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318572(2-{4-[6-Bromo-2-(4-dimethylaminomethylphenyl)-3H-i...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318594(6-Bromo-2-(4-methoxyphenyl)-7-[4-(5-methyl-isoxazo...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467119(CHEMBL4281827)
Affinity DataIC50:  17nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467118(CHEMBL4295199)
Affinity DataIC50:  17nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase C(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318596(3-((4-(6-Bromo-2-(4-(4-methylpiperazin-1-yl)phenyl...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant Aurora C expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318608(2-(4-(6-Chloro-7-(4-((5-methylisoxazol-3-yl)methyl...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381135(CHEMBL2017736)
Affinity DataIC50:  23nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318596(3-((4-(6-Bromo-2-(4-(4-methylpiperazin-1-yl)phenyl...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human recombinant Aurora B expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318607(2-(4-(6-Bromo-7-(4-((5-methylisoxazol-3-yl)methyl)...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318600(4-(4-(6-Bromo-7-(4-((1-methyl-1H-imidazol-2-yl)met...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318599(6-Bromo-2-(4-methoxyphenyl)-7-(4-((1-methyl-1H-imi...)
Affinity DataIC50:  32nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467120(CHEMBL4280027)
Affinity DataIC50:  33nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381134(CHEMBL2017735)
Affinity DataIC50:  39nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318591(6-Bromo-7-[4-(4-chlorobenzyl)-piperazin-1-yl]-2-(4...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381136(CHEMBL2017737)
Affinity DataIC50:  40nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50381139(CHEMBL2017871)
Affinity DataIC50:  40nMAssay Description:Inhibition of Mycobacterium tuberculosis GST-fused PknB expressed in Escherichia coli assessed as GarA substrate phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50224734(2-(4-(6-Chloro-2-(4-(dimethylamino)phenyl)-3H-imid...)
Affinity DataIC50:  42nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50224734(2-(4-(6-Chloro-2-(4-(dimethylamino)phenyl)-3H-imid...)
Affinity DataIC50:  42nMAssay Description:Inhibition of aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467115(CHEMBL4294776)
Affinity DataIC50:  47nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318569(2-(4-(6-Cyano-2-(4-(dimethylamino)phenyl)-3H-imida...)
Affinity DataIC50:  50nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50318574(2-(4-(6-Chloro-2-(4-methoxyphenyl)-3H-imidazo[4,5-...)
Affinity DataIC50:  52nMAssay Description:Inhibition of human recombinant Aurora A expressed in baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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