Affinity DataKi: 100nMAssay Description:Inhibition of [3H]dihydroalprenolol binding to Beta adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition of [3H]dihydroalprenolol binding to Beta adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of [3H]dihydroalprenolol binding to Beta adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of [3H]dihydroalprenolol binding to Beta adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of [3H]dihydroalprenolol binding to Beta adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of [3H]dihydroalprenolol binding to Beta adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Compounds were tested for inhibition against human liver Monoamine oxidase B (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of [3H]dihydroalprenolol binding to Beta adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of [3H]spiroperidol binding to dopamine receptor from rat striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of [3H]spiroperidol binding to dopamine receptor from rat striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Noncompetitive Inhibitory activity against rat striatal synaptosomal DHPR enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of [3H]spiroperidol binding to dopamine receptor from rat striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Binding affinity against Dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:Binding affinity against Dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 3.80E+3nMAssay Description:Inhibition of [3H]spiroperidol binding to dopamine receptor from rat striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Inhibition of [3H]dihydroalprenolol binding to Beta adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 4.50E+3nMAssay Description:Inhibition of [3H]spiroperidol binding to dopamine receptor from rat striatum membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 4.50E+3nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of [3H]spiroperidol binding to dopamine receptor from rat striatum membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of [3H]spiroperidol binding to dopamine receptor from rat striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 7.50E+3nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 7.50E+3nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Inhibition of [3H]spiroperidol binding to dopamine receptor from rat striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Compounds were tested for inhibition against human liver Monoamine oxidase B (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Compounds were tested for inhibition against human liver Monoamine oxidase B (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 1.70E+4nMAssay Description:Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 2.50E+4nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+4nMAssay Description:Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 2.70E+4nMAssay Description:Compound was tested for inhibition against human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 2.90E+4nMAssay Description:Compounds were tested for inhibition against human liver Monoamine oxidase B (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+4nMAssay Description:Inhibition of [3H]spiroperidol binding to dopamine receptor from rat striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+4nMAssay Description:Inhibition of [3H]dihydroalprenolol binding to Beta adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+4nMAssay Description:Inhibition of [3H]dihydroalprenolol binding to Beta adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+4nMAssay Description:Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 3.40E+4nMAssay Description:Inhibition of human placental Monoamine oxidase A (competitive inhibition was observed)More data for this Ligand-Target Pair
Affinity DataKi: 3.50E+4nMAssay Description:Inhibition of [3H]spiroperidol binding to dopamine receptor from rat striatum membranesMore data for this Ligand-Target Pair