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Found 262 with Last Name = 'brown' and Initial = 'je'
TargetHistamine H3 receptor(GUINEA PIG)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50071491(4-(1H-Imidazol-4-yl)-butyramidine | CHEMBL72156 | ...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of N-alpha-methylhistamine binding to histamine H3 receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  4.60nMAssay Description:Compound was evaluated for displacement of [3H]QNB from human Muscarinic m1 receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM81901(AF-DX 384 | CAS_119356 | CHEMBL279453 | NSC_119356)
Affinity DataKi:  5.30nMAssay Description:Compound was evaluated for displacement of [3H]-QNB from human Muscarinic m2 receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(GUINEA PIG)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50071496(CHEMBL73053 | N-(4-Chloro-benzyl)-2-[4-(1H-imidazo...)
Affinity DataKi:  7.20nMAssay Description:Inhibition of N-alpha-methylhistamine binding to histamine H3 receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  7.30nMAssay Description:Inhibition of N-alpha-methylhistamine binding to histamine H3 receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM81901(AF-DX 384 | CAS_119356 | CHEMBL279453 | NSC_119356)
Affinity DataKi:  12nMAssay Description:Compound was evaluated for displacement of [3H]QNB from human Muscarinic m1 receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023962(2-[(2,2-Dibromo-cyclopropanecarbonyl)-amino]-hex-2...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50071492(CHEMBL312341 | N-(4-Chloro-benzyl)-4-(1H-imidazol-...)
Affinity DataKi:  16nMAssay Description:Inhibition of N-alpha-methylhistamine binding to histamine H3 receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023979(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-7-(3...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024024(2-[(2,2-Dibromo-cyclopropanecarbonyl)-amino]-but-2...)
Affinity DataKi:  30nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50071488(4-(1H-Imidazol-4-ylmethyl)-benzamidine | CHEMBL736...)
Affinity DataKi:  38nMAssay Description:Inhibition of N-alpha-methylhistamine binding to histamine H3 receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023951(2-{6-Carboxy-6-[(2,2-dimethyl-cyclopropanecarbonyl...)
Affinity DataKi:  40nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024072(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-8-et...)
Affinity DataKi:  44nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023999(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hept...)
Affinity DataKi:  48nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  52nMAssay Description:Compound was evaluated for displacement of [3H]-QNB from human Muscarinic m2 receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024019(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-oct-...)
Affinity DataKi:  58nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024071(2-[(2,2-Dichloro-cyclopropanecarbonyl)-amino]-oct-...)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367508(CHEMBL1907817)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289120(4-Methyl-1-[2-oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyr...)
Affinity DataKi:  71nMAssay Description:Compound was evaluated for displacement of [3H]-QNB from human Muscarinic m2 receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023983(2-[(2,2-Dichloro-cyclopropanecarbonyl)-amino]-but-...)
Affinity DataKi:  80nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367506(CHEMBL1907823)
Affinity DataKi:  80nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289120(4-Methyl-1-[2-oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyr...)
Affinity DataKi:  82nMAssay Description:Compound was evaluated for displacement of [3H]QNB from human Muscarinic m1 receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023933(8-Cyano-2-[(2,2-dimethyl-cyclopropanecarbonyl)-ami...)
Affinity DataKi:  82nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024023(CHEMBL276215 | Sodium; 6-carboxy-6-[(2,2-dimethyl-...)
Affinity DataKi:  87nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024055(2-{6-Carboxy-6-[(2,2-dimethyl-cyclopropanecarbonyl...)
Affinity DataKi:  90nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023947(2,11-Bis-[(2,2-dimethyl-cyclopropanecarbonyl)-amin...)
Affinity DataKi:  92nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024044(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-dec-...)
Affinity DataKi:  96nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023992(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-7-ph...)
Affinity DataKi:  100nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023990(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hept...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023995(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-dode...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024045(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hex-...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367502(CILASTATIN)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024042(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-unde...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023942(10-Bromo-2-[(2,2-dimethyl-cyclopropanecarbonyl)-am...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024036(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-5-me...)
Affinity DataKi:  120nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024003(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-6-(3...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024069(7-Carboxymethylsulfanyl-2-[(2,2-dimethyl-cycloprop...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50071494(4-(1H-Imidazol-4-ylmethyl)-N-(4-trifluoromethyl-be...)
Affinity DataKi:  140nMAssay Description:Inhibition of N-alpha-methylhistamine binding to histamine H3 receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024078(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-trid...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023971(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hex-...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024059(7-Bromo-2-[(2,2-dimethyl-cyclopropanecarbonyl)-ami...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367507(CHEMBL1237318)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024012(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-8-me...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023946(4-Cyclohexyl-2-[(2,2-dimethyl-cyclopropanecarbonyl...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023963(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-6-me...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367505(CHEMBL1907816)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367509(CHEMBL1907822)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024058(7-(2-Carboxy-2-oxo-ethylsulfanyl)-2-[(2,2-dimethyl...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024053(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-7-me...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024066(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-non-...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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