Compile Data Set for Download or QSAR
maximum 50k data
Found 226 with Last Name = 'bruni' and Initial = 'b'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50428854(CHEMBL1236924)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma LBD expressed in HEK293 cells by filtration assayMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50002903(CHEMBL223836)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50002903(CHEMBL223836)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50417350(CHEMBL374584)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50417350(CHEMBL374584)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50085683((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2c receptor expressed in CHO cells in presence of GppNHp/NaChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50002904(CHEMBL222928)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50002905(CHEMBL373535)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50417341(CHEMBL397753)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50417354(CHEMBL396013)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50002905(CHEMBL373535)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50417353(CHEMBL242265)
Affinity DataKi:  186nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50002904(CHEMBL222928)
Affinity DataKi:  234nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataKi:  257nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50002903(CHEMBL223836)
Affinity DataKi:  269nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50417354(CHEMBL396013)
Affinity DataKi:  302nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50417350(CHEMBL374584)
Affinity DataKi:  355nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataKi:  363nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2c receptor expressed in CHO cells in presence of GppNHp/NaChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataKi:  501nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50417341(CHEMBL397753)
Affinity DataKi:  537nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50417354(CHEMBL396013)
Affinity DataKi:  589nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50002904(CHEMBL222928)
Affinity DataKi:  661nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataKi:  741nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50002905(CHEMBL373535)
Affinity DataKi:  933nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50417353(CHEMBL242265)
Affinity DataKi:  977nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50417353(CHEMBL242265)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50385682(CHEMBL390842)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50417341(CHEMBL397753)
Affinity DataKi:  1.59E+3nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50006584((McN-A-343) [4-(3-Chloro-phenylcarbamoyloxy)-but-2...)
Affinity DataKi:  1.95E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50006584((McN-A-343) [4-(3-Chloro-phenylcarbamoyloxy)-but-2...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50006584((McN-A-343) [4-(3-Chloro-phenylcarbamoyloxy)-but-2...)
Affinity DataKi:  3.24E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50006584((McN-A-343) [4-(3-Chloro-phenylcarbamoyloxy)-but-2...)
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50415218(CHEMBL404557)
Affinity DataKi:  4.90E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50385682(CHEMBL390842)
Affinity DataKi:  7.59E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50385682(CHEMBL390842)
Affinity DataKi:  7.76E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50006584((McN-A-343) [4-(3-Chloro-phenylcarbamoyloxy)-but-2...)
Affinity DataKi:  9.12E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50415225(CHEMBL593620)
Affinity DataKi:  1.05E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50415219(CHEMBL595265)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50415222(CHEMBL594376)
Affinity DataKi:  1.12E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50385682(CHEMBL390842)
Affinity DataKi:  1.15E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50415219(CHEMBL595265)
Affinity DataKi:  1.38E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50415219(CHEMBL595265)
Affinity DataKi:  1.55E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50415224(CHEMBL593685)
Affinity DataKi:  1.62E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50415215(CHEMBL593871)
Affinity DataKi:  1.66E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50415225(CHEMBL593620)
Affinity DataKi:  1.66E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 226 total ) | Next | Last >>
Jump to: