TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma LBD expressed in HEK293 cells by filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2c receptor expressed in CHO cells in presence of GppNHp/NaChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 186nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 234nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 257nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 269nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 302nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 355nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 363nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2c receptor expressed in CHO cells in presence of GppNHp/NaChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 537nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 589nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 661nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 741nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 933nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 977nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.23E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+3nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.59E+3nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.24E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.80E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.31E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 7.59E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 7.76E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.12E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.05E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.12E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.15E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.38E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.55E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.62E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.66E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.66E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair