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Found 185 with Last Name = 'campbell' and Initial = 'da'
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070256((R)-2-((S)-2-Hydroxy-3-mercapto-propyl)-nonanoic a...)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of matrix metalloproteinase-9, gelatinase-BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070257((R)-2-(3-Mercapto-2-oxo-propyl)-nonanoic acid ((S)...)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of matrix metalloproteinase-9, gelatinase-BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070228(2-(2-Mercapto-acetyl)-nonanoic acid ((S)-2,2-dimet...)
Affinity DataIC50:  0.300nMAssay Description:In vitro inhibitory activity against gelatinase-B(MMP-9).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070247(2-(2-Mercapto-acetyl)-nonanoic acid ((S)-2-cyclohe...)
Affinity DataIC50:  1.40nMAssay Description:In vitro inhibitory activity against gelatinase-B(MMP-9).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070227(2-(2-Mercapto-acetyl)-nonanoic acid ((S)-3-methyl-...)
Affinity DataIC50:  1.40nMAssay Description:In vitro inhibitory activity against gelatinase-B(MMP-9).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50070250(2-(1-Hydroxy-2-mercapto-ethyl)-5-phenyl-pentanoic ...)
Affinity DataIC50: >2nMAssay Description:In vitro inhibitory activity against stromelysin-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Phenomix

Curated by ChEMBL
LigandPNGBDBM50225074((1S,3S,5S)-2-[(S)-2-amino-2-(3-hydroxy-adamantan-1...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant DPP4 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Phenomix

Curated by ChEMBL
LigandPNGBDBM11695((2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}p...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant DPP4 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070226(2-(2-Mercapto-acetyl)-nonanoic acid {(S)-2-cyclohe...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibitory activity against gelatinase-B(MMP-9).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070256((R)-2-((S)-2-Hydroxy-3-mercapto-propyl)-nonanoic a...)
Affinity DataIC50:  5nMAssay Description:Inhibition of matrix metalloproteinase-1, Collagenase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50063920((R)-N*1*-((S)-2,2-Dimethyl-1-methylcarbamoyl-propy...)
Affinity DataIC50:  5nMAssay Description:Inhibition of matrix metalloproteinase-1, Collagenase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070223(2-(2-Mercapto-acetyl)-nonanoic acid ((S)-3-methyl-...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity against gelatinase-B(MMP-9).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070229(2-(2-Mercapto-acetyl)-4-methyl-pentanoic acid ((S)...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibitory activity against gelatinase-B(MMP-9).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070239(2-(2-Mercapto-acetyl)-nonanoic acid [(S)-3-methyl-...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibitory activity against gelatinase-B(MMP-9).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070253((2R,4S)-4-Hydroxy-2-isobutyl-5-mercapto-pentanoic ...)
Affinity DataIC50:  8nMAssay Description:Inhibition of matrix metalloproteinase-9, gelatinase-BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50070257((R)-2-(3-Mercapto-2-oxo-propyl)-nonanoic acid ((S)...)
Affinity DataIC50:  8nMAssay Description:Inhibition of matrix metalloproteinase-3, stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070254((R)-2-Isobutyl-5-mercapto-4-oxo-pentanoic acid ((S...)
Affinity DataIC50:  8nMAssay Description:Inhibition of matrix metalloproteinase-9, gelatinase-BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50070256((R)-2-((S)-2-Hydroxy-3-mercapto-propyl)-nonanoic a...)
Affinity DataIC50:  9nMAssay Description:Inhibition of matrix metalloproteinase-3, stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070235(2-(1-Hydroxy-2-mercapto-ethyl)-nonanoic acid [(S)-...)
Affinity DataIC50: >10nMAssay Description:In vitro inhibitory activity against collagenase-1(MMP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070257((R)-2-(3-Mercapto-2-oxo-propyl)-nonanoic acid ((S)...)
Affinity DataIC50:  10nMAssay Description:Inhibition of matrix metalloproteinase-1, Collagenase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070233(2-(1-Hydroxy-2-mercapto-ethyl)-nonanoic acid [(S)-...)
Affinity DataIC50: >10nMAssay Description:In vitro inhibitory activity against collagenase-1(MMP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070241(2-(2-Mercapto-acetyl)-nonanoic acid [(S)-1-(2-ethy...)
Affinity DataIC50: >10nMAssay Description:In vitro inhibitory activity against collagenase-1(MMP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070254((R)-2-Isobutyl-5-mercapto-4-oxo-pentanoic acid ((S...)
Affinity DataIC50:  11nMAssay Description:Inhibition of matrix metalloproteinase-1, Collagenase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070253((2R,4S)-4-Hydroxy-2-isobutyl-5-mercapto-pentanoic ...)
Affinity DataIC50:  11nMAssay Description:Inhibition of matrix metalloproteinase-1, Collagenase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50063920((R)-N*1*-((S)-2,2-Dimethyl-1-methylcarbamoyl-propy...)
Affinity DataIC50:  12nMAssay Description:Inhibition of matrix metalloproteinase-9, gelatinase-BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070251((R)-2-((R)-2-Hydroxy-3-mercapto-propyl)-nonanoic a...)
Affinity DataIC50:  12nMAssay Description:Inhibition of matrix metalloproteinase-9, gelatinase-BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50070240(2-(2-Mercapto-acetyl)-nonanoic acid [(S)-1-(2-ethy...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibitory activity against stromelysin-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070229(2-(2-Mercapto-acetyl)-4-methyl-pentanoic acid ((S)...)
Affinity DataIC50:  14nMAssay Description:In vitro inhibitory activity against collagenase-1(MMP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070228(2-(2-Mercapto-acetyl)-nonanoic acid ((S)-2,2-dimet...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibitory activity against collagenase-1(MMP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50070228(2-(2-Mercapto-acetyl)-nonanoic acid ((S)-2,2-dimet...)
Affinity DataIC50:  16nMAssay Description:In vitro inhibitory activity against stromelysin-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070234(2-(2-Mercapto-acetyl)-4-methyl-pentanoic acid [(S)...)
Affinity DataIC50:  19nMAssay Description:In vitro inhibitory activity against gelatinase-B(MMP-9).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50070225(2-(1-Hydroxy-2-mercapto-ethyl)-4-methyl-pentanoic ...)
Affinity DataIC50: >20nMAssay Description:In vitro inhibitory activity against stromelysin-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070258((R)-2-(3-Mercapto-2-oxo-propyl)-nonanoic acid [(S)...)
Affinity DataIC50:  20nMAssay Description:Inhibition of matrix metalloproteinase-9, gelatinase-BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070230(2-(1-Hydroxy-2-mercapto-ethyl)-nonanoic acid ((S)-...)
Affinity DataIC50: >20nMAssay Description:In vitro inhibitory activity against collagenase-1(MMP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070223(2-(2-Mercapto-acetyl)-nonanoic acid ((S)-3-methyl-...)
Affinity DataIC50: >20nMAssay Description:In vitro inhibitory activity against collagenase-1(MMP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070244(2-(1-Hydroxy-2-mercapto-ethyl)-nonanoic acid [(S)-...)
Affinity DataIC50: >20nMAssay Description:In vitro inhibitory activity against collagenase-1(MMP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50076153(2-((2S,5R)-2-(4-nitrobenzyl)-5-(mercaptomethyl)-3,...)
Affinity DataIC50:  21nMAssay Description:Inhibitory activity against Matrix metalloprotease-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50070236(2-(2-Mercapto-acetyl)-nonanoic acid {(S)-2,2-dimet...)
Affinity DataIC50:  22nMAssay Description:In vitro inhibitory activity against stromelysin-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50076158(2-((2S,5R)-2-(4-nitrobenzyl)-5-(mercaptomethyl)-3,...)
Affinity DataIC50:  24nMAssay Description:Inhibitory activity against Matrix metalloprotease-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070255((R)-2-((S)-2-Hydroxy-3-mercapto-propyl)-nonanoic a...)
Affinity DataIC50:  24nMAssay Description:Inhibition of matrix metalloproteinase-9, gelatinase-BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50076151(2-((2S,5R)-2-(4-nitrobenzyl)-5-(mercaptomethyl)-3,...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against Matrix metalloprotease-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50070241(2-(2-Mercapto-acetyl)-nonanoic acid [(S)-1-(2-ethy...)
Affinity DataIC50:  26nMAssay Description:In vitro inhibitory activity against stromelysin-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Phenomix

Curated by ChEMBL
LigandPNGBDBM50295970((3R,6S,7aS)-6-amino-5-oxo-6-phenylhexahydropyrrolo...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant DPP4 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50070242(2-(2-Mercapto-acetyl)-nonanoic acid [(S)-1-(2-ethy...)
Affinity DataIC50:  28nMAssay Description:In vitro inhibitory activity against stromelysin-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50064797((3R,6S)-6-Cyclohexylmethyl-3-mercaptomethyl-1-(4-m...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against Matrix metalloprotease-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50064797((3R,6S)-6-Cyclohexylmethyl-3-mercaptomethyl-1-(4-m...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Matrix Metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50070241(2-(2-Mercapto-acetyl)-nonanoic acid [(S)-1-(2-ethy...)
Affinity DataIC50:  30nMAssay Description:In vitro inhibitory activity against gelatinase-B(MMP-9).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Phenomix

Curated by ChEMBL
LigandPNGBDBM50295972((3R,6S,7aS)-6-amino-6-isopropyl-5-oxohexahydropyrr...)
Affinity DataIC50:  33nMAssay Description:Inhibition of human recombinant DPP4 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50064794((3R,6S)-6-Cyclohexylmethyl-3-mercaptomethyl-1-quin...)
Affinity DataIC50:  35nMAssay Description:Inhibition of Matrix Metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50076152(2-((2S,5R)-2-(4-nitrobenzyl)-5-(mercaptomethyl)-3,...)
Affinity DataIC50:  36nMAssay Description:Inhibitory activity against Matrix metalloprotease-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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