Affinity DataKi: 0.700nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 0.730nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Weizmann Institute Of Science
Weizmann Institute Of Science
Affinity DataKi: 0.800nM ΔG°: -51.4kJ/mole IC50: 2.40nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Weizmann Institute Of Science
Weizmann Institute Of Science
Affinity DataKi: 4.5nM ΔG°: -47.2kJ/mole IC50: 16nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Inhibition of [3H]- DA reuptake into rat striatal synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of [3H]- DA reuptake into rat striatal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 19.6nM ΔG°: -43.6kJ/mole IC50: 52nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 47.1nM ΔG°: -41.4kJ/mole IC50: 114nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of [3H]- DA reuptake into rat striatal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Inhibition of [3H]- DA reuptake into rat striatal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 137nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 143nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 164nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Weizmann Institute Of Science
Weizmann Institute Of Science
Affinity DataKi: 175nM ΔG°: -38.2kJ/mole IC50: 414nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Inhibition of [3H]- DA reuptake into rat striatal synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 360nMAssay Description:Inhibition of [3H]- DA reuptake into rat striatal synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 570nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 640nMAssay Description:Inhibition of [3H]- DA reuptake into rat striatal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 643nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Inhibition of [3H]5-HT reuptake into rat frontal cortex synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 830nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 990nMAssay Description:Inhibition of [3H]- NE reuptake into rat hippocampal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of [3H]- DA reuptake into rat striatal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition of [3H]- DA reuptake into rat striatal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.46E+3nMAssay Description:Inhibition of [3H]- DA reuptake into rat striatal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.55E+3nMAssay Description:Inhibition of [3H]- DA reuptake into rat striatal synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Hong Kong University Of Science And Technology
Curated by ChEMBL
Hong Kong University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of [3H]- DA reuptake into rat striatal synaptosomesMore data for this Ligand-Target Pair