Affinity DataKi: 3.5nMAssay Description:Inhibition of human erythrocytes BChEMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibition of human plasma BChEMore data for this Ligand-Target Pair
Affinity DataKi: 8.60nMAssay Description:Mixed-type reversible inhibition of bovine acetylcholinesterase using S-acetylthiocholine as substrate incubated for 20 mins prior to substrate addit...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Competitive inhibition of human recombinant MAO-B expressed in supersomes using kynuramine as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Inhibition of bovine AChE at 30 nM using S-acetylthiocholine as as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Mixed/noncompetitive inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addi...More data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Mixed/noncompetitive inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addi...More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Mixed type inhibition of electric eel AChE by Lineweaver-Burk plotMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataKi: 93nMAssay Description:Binding affinity to recombinant human MAO-B expressed in Pichia pastoris assessed as inhibition constant using benzylamine as substrate by Michaelis-...More data for this Ligand-Target Pair
Affinity DataKi: 93.4nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholineiodide as substrate measured for every 30 sec for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Mixed type inhibition of equine serum BChE assessed as Ki using butyrylthiocholine as substrate preincubated for 20 mins followed by substrate additi...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Mixed type inhibition of electric eel AChE by Lineweaver-Burk plotMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Binding affinity to recombinant human MAO-B expressed in Pichia pastoris assessed as inhibition constant using benzylamine as substrate by Michaelis-...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:Binding affinity to recombinant human MAO-B expressed in Pichia pastoris assessed as inhibition constant using benzylamine as substrate by Michaelis-...More data for this Ligand-Target Pair
Affinity DataKi: 1.37E+3nMAssay Description:Mixed-type inhibition of electric eel AChE using S-acetylthiocholine as substrate preincubated for 20 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
Affinity DataKi: 1.37E+3nMAssay Description:Mixed-type inhibition of electric eel AChE using S-acetylthiocholine as substrate preincubated for 20 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Mixed type inhibition of human AChE by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataKi: 4.50E+3nMAssay Description:Tight binding inhibition of recombinant human MAO-B expressed in Pichia pastoris assessed as inhibition constant using benzylamine as substrate at 10...More data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Inhibition of bovine AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Inhibition of bovine AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Inhibition of bovine AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human recombinant AChE using ATCh as substrate preincubated for 20 mins followed by substrate addition and measured for 3 mins by Ellma...More data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human AChE by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 0.912nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 0.912nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of bovine AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetCytochrome P450 11B2, mitochondrial(Homo sapiens (Human))
Universita` Degli Studi Di Bari Aldo Moro
Curated by ChEMBL
Universita` Degli Studi Di Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of human CYP11B2 expressed in Chinese hamster V79MZ cells using [1,2-3H]11-deoxycorticosterone/11-deoxycorticosteroneMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.07nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against monoamine oxidase BMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.12nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.12nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
Affinity DataIC50: 1.15nMAssay Description:Inhibitory effect on Monoamine oxidase B, SD on IC50 values < 10%More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.38nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.38nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.41nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.48nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.55nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.58nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.62nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.66nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.78nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Bari "Aldo Moro
Curated by ChEMBL
University Of Bari "Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.95nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of acetylcholinesterase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of bovine AChE by Ellman's methodMore data for this Ligand-Target Pair