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Found 129 with Last Name = 'compain' and Initial = 'p'
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50315250((2R,3S,4S,5R)-2-nonylpiperidine-3,4,5-triol | CHEM...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of human recombinant beta-glucocerebrosidase assessed as p-nitrophenolate accumulation preincubated for 10 mins before p-nitrophenyl-beta-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM18364((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-nonylpiperidi...)
Affinity DataKi:  200nM ΔG°:  -39.8kJ/mole IC50:  270nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM18363((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-octylpiperidi...)
Affinity DataKi:  280nM ΔG°:  -38.9kJ/mole IC50:  500nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM18358((2R,3R,4R,5S)-2-(hydroxymethyl)-1-nonylpiperidine-...)
Affinity DataKi:  300nM ΔG°:  -38.7kJ/mole IC50:  660nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM18357((2R,3R,4R,5S)-2-(hydroxymethyl)-1-octylpiperidine-...)
Affinity DataKi:  420nM ΔG°:  -37.9kJ/mole IC50:  820nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM18362((2R,3S,4R,5R,6R)-2-hexyl-6-(hydroxymethyl)piperidi...)
Affinity DataKi:  2.30E+3nM ΔG°:  -33.5kJ/mole IC50:  4.20E+3nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM18356((2R,3R,4R,5S)-1-hexyl-2-(hydroxymethyl)piperidine-...)
Affinity DataKi:  5.50E+3nM ΔG°:  -31.2kJ/mole IC50:  1.30E+4nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  7.90E+4nM ΔG°:  -24.4kJ/mole IC50:  2.40E+5nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM18361((2R,3S,4R,5R,6R)-2-butyl-6-(hydroxymethyl)piperidi...)
Affinity DataKi:  1.10E+5nM ΔG°:  -23.5kJ/mole IC50:  1.00E+5nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM18355((2R,3R,4R,5S)-1-butyl-2-(hydroxymethyl)piperidine-...)
Affinity DataKi:  1.16E+5nM ΔG°:  -23.4kJ/mole IC50:  2.70E+5nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156360(2-Hydroxymethyl-6-nonyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50315255((2R,3S,4S,5R)-2-hexylpiperidine-3,4,5-triol | CHEM...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant beta-glucocerebrosidase assessed as p-nitrophenolate accumulation preincubated for 10 mins before p-nitrophenyl-beta-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral alpha-glucosidase C(Homo sapiens (Human))
Institut De Chimie Organique Et Analytique (I.C.O.A.)

Curated by ChEMBL
LigandPNGBDBM50082234((3R,4R,5S)-2,6-Bis-hydroxymethyl-piperidine-3,4,5-...)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against alpha-galactosidase from coffee bean.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative alpha-glucosidase(Oryza sativa subsp. japonica)
Universit£

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against alpha-Glucosidase from riceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  73nMAssay Description:Inhibition of human recombinant serum BuchE using butyrylthiocholine iodide as substrate by Ellman methodMore data for this Ligand-Target Pair
TargetPutative alpha-glucosidase(Oryza sativa subsp. japonica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156357(2-Hydroxymethyl-1-nonyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  80nMAssay Description:Inhibitory activity against alpha-Glucosidase from riceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative alpha-glucosidase(Oryza sativa subsp. japonica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156359(2-Hydroxymethyl-1-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  80nMAssay Description:Inhibitory activity against alpha-Glucosidase from riceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156356(2-Hydroxymethyl-6-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  90nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  136nMAssay Description:Inhibition of electric eel AchE using acetylthiocholine iodide as substrate by Ellman methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156355(2-Butyl-6-hydroxymethyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  150nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50:  210nMAssay Description:Inhibitory activity against rat intestinal sucrase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156357(2-Hydroxymethyl-1-nonyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  230nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156359(2-Hydroxymethyl-1-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  280nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50:  300nMAssay Description:Inhibitory activity against rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156353(2-Hexyl-6-hydroxymethyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  310nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral alpha-glucosidase C(Mus musculus)
Institut De Chimie Organique Et Analytique (I.C.O.A.)

Curated by ChEMBL
LigandPNGBDBM50259956(2,6-Bis-hydroxymethyl-piperidine-3,4,5-triol | CHE...)
Affinity DataIC50:  340nMAssay Description:Inhibitory activity against alpha-glucosidase from rat intestinal maltaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50:  360nMAssay Description:Inhibitory activity against rat intestinal maltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative alpha-glucosidase(Oryza sativa subsp. japonica)
Universit£

Curated by ChEMBL
LigandPNGBDBM18355((2R,3R,4R,5S)-1-butyl-2-(hydroxymethyl)piperidine-...)
Affinity DataIC50:  420nMAssay Description:Inhibitory activity against alpha-Glucosidase from riceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156354(1-Hexyl-2-hydroxymethyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  450nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156354(1-Hexyl-2-hydroxymethyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  450nMAssay Description:Inhibition of rat intestinal sucrase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  484nMAssay Description:Inhibition of human recombinant AchE using acetylthiocholine iodide as substrate by Ellman methodMore data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156358(2-Hydroxymethyl-6-propyl-piperidine-3,4,5-triol | ...)
Affinity DataIC50:  530nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50315252((2R,3S,4S,5R)-2-propylpiperidine-3,4,5-triol | CHE...)
Affinity DataIC50:  560nMAssay Description:Inhibition of human recombinant beta-glucocerebrosidase assessed as p-nitrophenolate accumulation preincubated for 10 mins before p-nitrophenyl-beta-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative alpha-glucosidase(Oryza sativa subsp. japonica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156356(2-Hydroxymethyl-6-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  590nMAssay Description:Inhibitory activity against alpha-Glucosidase from riceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156357(2-Hydroxymethyl-1-nonyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  660nMAssay Description:Inhibition of rat intestinal sucrase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156359(2-Hydroxymethyl-1-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  660nMAssay Description:Inhibition of rat intestinal sucrase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative alpha-glucosidase(Oryza sativa subsp. japonica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156354(1-Hexyl-2-hydroxymethyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against alpha-Glucosidase from riceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative alpha-glucosidase(Oryza sativa subsp. japonica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156353(2-Hexyl-6-hydroxymethyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  800nMAssay Description:Inhibitory activity against alpha-Glucosidase from riceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
Hokuriku University

LigandPNGBDBM18353((2R,3R,4R,5S)-2-(hydroxymethyl)-1-methylpiperidine...)
Affinity DataIC50:  1.00E+3nMpH: 4.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
Hokuriku University

LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataIC50:  1.00E+3nMpH: 4.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
Hokuriku University

LigandPNGBDBM18366((2R,3R,5S,6R)-2,6-bis(hydroxymethyl)piperidine-3,4...)
Affinity DataIC50:  1.00E+3nMpH: 4.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50061158(CHEMBL3393676)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human recombinant serum BuchE using butyrylthiocholine iodide as substrate by Ellman methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156353(2-Hexyl-6-hydroxymethyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of rat intestinal sucrase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156357(2-Hydroxymethyl-1-nonyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of rat intestinal maltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156361(2-Hydroxymethyl-1-propyl-piperidine-3,4,5-triol | ...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156356(2-Hydroxymethyl-6-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rat intestinal sucrase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156359(2-Hydroxymethyl-1-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rat intestinal maltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
Hokuriku University

LigandPNGBDBM18358((2R,3R,4R,5S)-2-(hydroxymethyl)-1-nonylpiperidine-...)
Affinity DataIC50:  1.50E+3nMpH: 4.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative alpha-glucosidase(Oryza sativa subsp. japonica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156360(2-Hydroxymethyl-6-nonyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity against alpha-Glucosidase from riceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156356(2-Hydroxymethyl-6-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of rat intestinal maltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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