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Found 21 with Last Name = 'coudert' and Initial = 'g'
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50260343(10-Hydroxy-1H-pyrido[3'4':4,5]pyrrolo[2,3-a]pyrrol...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human Chk1 expressed in sf9-baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50260341(10-Benzyloxy-1H-pyrido[3'4':4,5]pyrrolo[2,3-a]-pyr...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human Chk1 expressed in sf9-baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50260358(9-Hydroxy-1H-pyrido[3'4':4,5]pyrrolo[2,3-a]pyrrolo...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human Chk1 expressed in sf9-baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50260340(9-Benzyloxy-1H-pyrido[3'4':4,5]pyrrolo[2,3-a]pyrro...)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibition of human Chk1 expressed in sf9-baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50260334(10-Hydroxy-6-methyl-1H-pyrido[3'4':4,5]pyrrolo-[2,...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human Chk1 expressed in sf9-baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50260339(1H-pyrido[3'4':4,5]pyrrolo[2,3-a]pyrrolo[3,4-c]-ca...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human Chk1 expressed in sf9-baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404697(CHEMBL174882)
Affinity DataKd:  617nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404698(CHEMBL366558)
Affinity DataKd:  1.18E+3nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404696(CHEMBL427310)
Affinity DataKd:  8.5nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404696(CHEMBL427310)
Affinity DataKd:  81.3nMAssay Description:Antagonist activity of compound against Beta-2 adrenergic receptor in isolated guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKd:  43.6nMAssay Description:Antagonist activity of compound against Beta-2 adrenergic receptor in isolated guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404697(CHEMBL174882)
Affinity DataKd:  1.35E+3nMAssay Description:Antagonist activity of compound against Beta-2 adrenergic receptor in isolated guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404698(CHEMBL366558)
Affinity DataKd:  1.70E+4nMAssay Description:Antagonist activity of compound against Beta-2 adrenergic receptor in isolated guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404699(CHEMBL175010)
Affinity DataKd:  162nMAssay Description:Antagonist activity of compound against Beta-2 adrenergic receptor in isolated guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404695(CHEMBL174853)
Affinity DataKd:  2nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKd:  8.70nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM25749(CHEMBL6995 | N-{4-[2-hydroxy-3-(propan-2-ylamino)p...)
Affinity DataKd:  174nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404700(CHEMBL360139)
Affinity DataKd:  145nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404695(CHEMBL174853)
Affinity DataKd:  178nMAssay Description:Antagonist activity of compound against Beta-2 adrenergic receptor in isolated guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404694(CHEMBL173882)
Affinity DataKd:  263nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404699(CHEMBL175010)
Affinity DataKd:  15nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed