Affinity DataKi: 0.200nMAssay Description:Agonist activity at recombinant human full length CB2 receptor expressed in HEK293 cell membranes after 2 hrs by [35S]GTP-gammaS binding assayMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 0.470nMAssay Description:Displacement of [3H]EYF from human NPFF2 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]CP-55,940 from recombinant human full length CB1 receptor expressed in HEK293 cell membranes after 90 mins by topcount methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Displacement of [3H]CP-55,940 from recombinant human full length CB2 receptor expressed in HEK293 cell membranes after 90 mins by topcount methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Agonist activity at recombinant human full length CB1 receptor expressed in HEK293 cell membranes after 2 hrs by [35S]GTP-gammaS binding assayMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [125I]EYF from human NPFF2 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [125I]YVP from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 4.80nMAssay Description:Displacement of [3H]U-69593 from human KOR expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Displacement of [3H]CP-55,940 from recombinant human full length CB2 receptor expressed in HEK293 cell membranes after 90 mins by topcount methodMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor (unknown origin) transfected into HEK293 cells by microplate scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]EYF from human NPFF2 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Agonist activity at recombinant human full length CB1 receptor expressed in HEK293 cell membranes after 2 hrs by [35S]GTP-gammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Displacement of [3H]CP-55,940 from recombinant human full length CB1 receptor expressed in HEK293 cell membranes after 90 mins by topcount methodMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Agonist activity at recombinant human full length CB1 receptor expressed in HEK293 cell membranes after 2 hrs by [35S]GTP-gammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Competitive inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinoline formation using varying levels of kynuramine as substra...More data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Antagonist activity at human NPFF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Competitive inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinoline formation using varying levels of kynuramine as substra...More data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 75nMAssay Description:Antagonist activity at human NPFF2 receptor expressed in African green monkey COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Displacement of [3H]EYF from human NPFF2 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 84nMAssay Description:Displacement of [3H]EYF from human NPFF2 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 94nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 114nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 117nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
Affinity DataKi: 124nMAssay Description:Mixed-type inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinoline formation using varying levels of kynuramine as substrat...More data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 129nMAssay Description:Displacement of [3H]EYF from human NPFF2 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 129nMAssay Description:Displacement of [3H]CP55940 from full length human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
Affinity DataKi: 137nMAssay Description:Displacement of [3H]CP-55,940 from recombinant human full length CB1 receptor expressed in HEK293 cell membranes after 90 mins by topcount methodMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 141nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 151nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Displacement of [3H]CP-55,940 from recombinant human full length CB2 receptor expressed in HEK293 cell membranes after 90 mins by topcount methodMore data for this Ligand-Target Pair
Affinity DataKi: 163nMAssay Description:Mixed-type inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinoline formation using varying levels of kynuramine as substrat...More data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 191nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 193nMAssay Description:Agonist activity at recombinant human full length CB1 receptor expressed in HEK293 cell membranes after 2 hrs by [35S]GTP-gammaS binding assayMore data for this Ligand-Target Pair
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 201nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair