TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: >0.0480nMAssay Description:Binding affinity to human adenosine A2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Binding affinity at adenosine A2A receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Binding affinity at adenosine A2A receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Binding affinity at adenosine A2A receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity at adenosine A2A receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair