TargetEstrogen receptor(Mus musculus)
University Of New Mexico Health Sciences Center
Curated by ChEMBL
University Of New Mexico Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Binding affinity to ERalpha receptor in mouse COS7 cells by competitive binding assayMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Mus musculus)
University Of New Mexico Health Sciences Center
Curated by ChEMBL
University Of New Mexico Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Binding affinity to ERbeta receptor in mouse COS7 cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >0.300nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
New Mexico State University
Curated by ChEMBL
New Mexico State University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Binding affinity to GPR30More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of specific binding of [125-I] ET-1 to human Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of the specific binding of [125I]-angiotensin II to a guinea pig adrenal membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:In vitro inhibition of the specific binding of [125I]-angiotensin II to a guinea pig adrenal membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:In vitro inhibition of the specific binding of [125I]-angiotensin II to a guinea pig adrenal membrane preparationMore data for this Ligand-Target Pair
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
New Mexico State University
Curated by ChEMBL
New Mexico State University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Binding affinity to GPR30More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:In vitro inhibition of the specific binding of [125I]-angiotensin II to a guinea pig adrenal membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:In vitro inhibition of the specific binding of [125I]-angiotensin II to a guinea pig adrenal membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:In vitro inhibition of the specific binding of [125I]-angiotensin II to a guinea pig adrenal membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:In vitro inhibition of the specific binding of [125I]-angiotensin II to a guinea pig adrenal membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of the specific binding of [125I]-angiotensin II to a guinea pig adrenal membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair