Affinity DataKi: 0.000800nMAssay Description:Binding affinity towards Wild-type kappa opioid receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0240nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Displacement of [3H]diprenorphine from opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0890nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Displacement of [3H]- diprenorphine from delta receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.214nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 0.226nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]diprenorphine from delta-W284E-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.244nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 0.354nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Displacement of [3H]- diprenorphine from mu-W318A-receptor expressed in HEK 293More data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Displacement of [3H]- diprenorphine from mu-W318A-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Displacement of [3H]- diprenorphine from mu-W318A-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.529nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding constant against E203Q,D204N,D206N EL-2 Opioid receptor kappa 1 using [3H]diprenorphine as radioligand expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding constant against wild type EL-2 Opioid receptor kappa 1 using [3H]diprenorphine as radioligand expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.823nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding constant against E203Q,D204N,D206N,E209Q EL-2 Opioid receptor kappa 1 using [3H]diprenorphine as radioligand expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.13nMAssay Description:Effect on binding to wild-type opioid receptor kappa 1 using [3H]diprenorphine in transiently expressed rat HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.15nMAssay Description:Binding affinity towards rat opioid receptor kappa 1 was determined using [3H]diprenorphine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.23nMAssay Description:Displacement of [3H]diprenorphine from k-Y312A-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.39nMAssay Description:Displacement of [3H]diprenorphine from k-Y312A-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.82nMAssay Description:Displacement of [3H]- diprenorphine from delta-W284E-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity towards delta-opioid receptor from CHO cellsMore data for this Ligand-Target Pair
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Inhibition of Mycobacterium tuberculosis BAG RV143 MbtA expressed in Escherichia coli BL21 (DE3) assessed as ATP-[32P]PPi exchange by liquid scintill...More data for this Ligand-Target Pair
Affinity DataKi: 2.75nMAssay Description:Binding affinity towards mouse delta-opioid receptor was determined using [3H]diprenorphine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.83nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Inhibition of Mycobacterium tuberculosis BAG RV143 MbtA expressed in Escherichia coli BL21 (DE3) assessed as ATP-[32P]PPi exchange by liquid scintill...More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity against Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Binding constant against D216N,D217N,E218Q EL-2 Opioid receptor kappa 1 using [3H]diprenorphine as radioligand expressed in HEK cellsMore data for this Ligand-Target Pair
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Inhibition of Mycobacterium tuberculosis BAG RV143 MbtA expressed in Escherichia coli BL21 (DE3) assessed as ATP-[32P]PPi exchange by liquid scintill...More data for this Ligand-Target Pair
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Inhibition of Mycobacterium tuberculosis BAG RV143 MbtA expressed in Escherichia coli BL21 (DE3) assessed as ATP-[32P]PPi exchange by liquid scintill...More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]- diprenorphine from mu-W318A-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]- diprenorphine from delta receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.46nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Inhibition of Mycobacterium tuberculosis BAG RV143 MbtA expressed in Escherichia coli BL21 (DE3) assessed as ATP-[32P]PPi exchange by liquid scintill...More data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Displacement of [3H]- diprenorphine from delta-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.46nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 12.3nMAssay Description:Effect on binding to kappa(Glu297Ala) opioid receptor, using [3H]diprenorphine in transiently expressed rat HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12.8nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 13.5nMAssay Description:Displacement of [3H]- diprenorphine from mu-K303E-receptor expressed in HEK 293More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity towards mu-opioid receptor from CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 15.7nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 17.4nMAssay Description:Displacement of [3H]- diprenorphine from mu-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17.5nMAssay Description:Displacement of [3H]diprenorphine from rat kappa opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity towards opioid receptor kappa 1 from CHO cellsMore data for this Ligand-Target Pair