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Found 239 with Last Name = 'fisher' and Initial = 'rj'
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362892(CHEMBL1946564)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of FITC-conjugated (S)-4-((S)-1-acetylpyrrolidine-2-carboxamido)-5-((2S,4R)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-((S)-1-((S)-1-amino-4-carb...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362891(CHEMBL1946260)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of FITC-conjugated (S)-4-((S)-1-acetylpyrrolidine-2-carboxamido)-5-((2S,4R)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-((S)-1-((S)-1-amino-4-carb...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362890(CHEMBL1946259)
Affinity DataKi:  5.40E+3nMAssay Description:Displacement of FITC-conjugated (S)-4-((S)-1-acetylpyrrolidine-2-carboxamido)-5-((2S,4R)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-((S)-1-((S)-1-amino-4-carb...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362889(CHEMBL1946129)
Affinity DataKi:  8.70E+3nMAssay Description:Displacement of FITC-conjugated (S)-4-((S)-1-acetylpyrrolidine-2-carboxamido)-5-((2S,4R)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-((S)-1-((S)-1-amino-4-carb...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50139763(CHEMBL306657 | [(E)-(9S,10S,14S,18S)-18-Carbamoylm...)
Affinity DataIC50:  1.40nMAssay Description:In vitro Growth factor receptor bound protein 2-binding affinity of the compound was determined in in surface plasmon resonance (SPR) methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50139763(CHEMBL306657 | [(E)-(9S,10S,14S,18S)-18-Carbamoylm...)
Affinity DataIC50:  1.40nMAssay Description:In vitro Growth factor receptor bound protein 2-binding affinity of the compound was determined in in surface plasmon resonance (SPR) methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50139763(CHEMBL306657 | [(E)-(9S,10S,14S,18S)-18-Carbamoylm...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity in extracellular ELISA-based assay for Grb2 SH2 domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50168312(2-{4-[(16R,20S)-18-((S)-Carbamoylmethyl)-9-carboxy...)
Affinity DataIC50:  3.30nMAssay Description:Inhibitory concentration against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50143944(2-[4-((E)-(9S,10S,14S,18S)-18-Carbamoylmethyl-9-ca...)
Affinity DataIC50:  4.30nMAssay Description:In vitro Growth factor receptor bound protein 2-binding affinity of the compound was determined in ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50168318(CHEMBL424823 | [(15R,20S)-18-Carbamoylmethyl-10-[4...)
Affinity DataIC50:  6.30nMAssay Description:Inhibitory concentration against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50168317(CHEMBL193281 | [(15R,20S)-10-[4-(Benzyl-hydroxy-ph...)
Affinity DataIC50:  8.40nMAssay Description:Inhibitory concentration against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50168316(CHEMBL263328 | N-{4-[(7S,14R,18S)-18-Carbamoylmeth...)
Affinity DataIC50:  8.80nMAssay Description:Inhibitory concentration against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50072865(CHEMBL55627 | N-[(S)-1-{1-[(S)-2-Carbamoyl-1-(3-na...)
Affinity DataIC50:  10nMAssay Description:In vitro Growth factor receptor bound protein 2-binding affinity of the compound was determined in ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50143944(2-[4-((E)-(9S,10S,14S,18S)-18-Carbamoylmethyl-9-ca...)
Affinity DataIC50:  12.1nMAssay Description:In vitro Growth factor receptor bound protein 2-binding affinity of the compound was determined in in surface plasmon resonance (SPR) methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50139762(CHEMBL349373 | [(16R,20S)-18-((S)-Carbamoylmethyl)...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50102025(4-[(10S,14S,18S)-18-(2-AMINO-2-OXOETHYL)-14-(1-NAP...)
Affinity DataIC50:  20nMAssay Description:In vitro binding affinity in extracellular ELISA-based assay for Grb2 SH2 domainMore data for this Ligand-Target Pair
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50085867(2-(4-((S)-3-(1-((S)-4-amino-1-(3-(naphthalen-1-yl)...)
Affinity DataIC50:  22.1nMAssay Description:In vitro Growth factor receptor bound protein 2-binding affinity of the compound was determined in ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50168314(CHEMBL193015 | [(7S,14R,18S)-18-Carbamoylmethyl-10...)
Affinity DataIC50:  22.5nMAssay Description:Inhibitory concentration against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50072862(CHEMBL117807 | Phosphoric acid mono-[4-((S)-2-acet...)
Affinity DataIC50:  47nMAssay Description:Inhibition of Grb2 SH2 domain binding in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50085867(2-(4-((S)-3-(1-((S)-4-amino-1-(3-(naphthalen-1-yl)...)
Affinity DataIC50:  70nMAssay Description:Inhibition of Grb2 SH2 domain binding in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50161466((R)-N-(1-{(S)-2-Carbamoyl-1-[2-(7-nitro-benzo[1,2,...)
Affinity DataIC50:  167nMAssay Description:Apparent dissociation constant for human growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50085877(CHEMBL355066 | N-[(S)-1-{1-[(S)-2-Carbamoyl-1-(3-n...)
Affinity DataIC50:  600nMAssay Description:Inhibition of Grb2 SH2 domain bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50085877(CHEMBL355066 | N-[(S)-1-{1-[(S)-2-Carbamoyl-1-(3-n...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Grb2 SH2 domain binding in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSHC-transforming protein 1(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50276388(4-((S)-2-acetamido-3-((S)-5-amino-1-((2-((S)-1-ami...)
Affinity DataIC50:  6.00E+3nMAssay Description:Displacement of FITC-tagged NH-(CH2)4-CO-phospho-tyrosine-glutamine-glycine-leucine-serine-amide from Shc Src homology 2 domain (unknown origin) by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50158383(2-((8S,9S,10R,13S,14S,17S)-10,13-dimethyl-3-oxo-2,...)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of human Tdp1 expressed in Escherichia coli assessed as blockade of enzyme-mediated hydrolysis of phosphodiester linkage between tyrosine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSHC-transforming protein 1(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50276339(4-((2S,5S,11S,14S)-2-acetamido-5-(3-amino-3-oxopro...)
Affinity DataIC50:  8.00E+3nMAssay Description:Displacement of FITC-tagged NH-(CH2)4-CO-phospho-tyrosine-glutamine-glycine-leucine-serine-amide from Shc Src homology 2 domain (unknown origin) by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSHC-transforming protein 1(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50276387(4-((S)-2-acetamido-3-((S)-5-amino-1-((2-((S)-1-ami...)
Affinity DataIC50:  8.90E+3nMAssay Description:Displacement of FITC-tagged NH-(CH2)4-CO-phospho-tyrosine-glutamine-glycine-leucine-serine-amide from Shc Src homology 2 domain (unknown origin) by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSHC-transforming protein 1(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50276396(4-((S)-2-acetamido-3-((S)-5-amino-1-((2-((S)-1-ami...)
Affinity DataIC50:  1.00E+4nMAssay Description:Displacement of FITC-tagged NH-(CH2)4-CO-phospho-tyrosine-glutamine-glycine-leucine-serine-amide from Shc Src homology 2 domain (unknown origin) by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230460(5-[(1Z)-({[(2S,3S)-2-{[(1S)-1-{[(1S)-1-carbamoyl-3...)
Affinity DataIC50:  1.10E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230470((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.20E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362891(CHEMBL1946260)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human Tsg101 binding to GST-tagged P6 protein by surface plasmon resonance methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230449((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.20E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230450(4-carbamoyl-4-(4-carboxy-2-{[(2S,3S)-1-({1-[(2S)-2...)
Affinity DataIC50:  1.20E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50371256(CHEMBL1162967)
Affinity DataIC50:  1.30E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230469((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.30E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSHC-transforming protein 1(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50276402(4-((S)-2-acetamido-3-((S)-5-amino-1-((2-((S)-1-ami...)
Affinity DataIC50:  1.40E+4nMAssay Description:Displacement of FITC-tagged NH-(CH2)4-CO-phospho-tyrosine-glutamine-glycine-leucine-serine-amide from Shc Src homology 2 domain (unknown origin) by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSHC-transforming protein 1(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50276346(4-((2S,5S,11S)-2-acetamido-5-(3-amino-3-oxopropyl)...)
Affinity DataIC50:  1.40E+4nMAssay Description:Displacement of FITC-tagged NH-(CH2)4-CO-phospho-tyrosine-glutamine-glycine-leucine-serine-amide from Shc Src homology 2 domain (unknown origin) by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230462((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.50E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50124303(3-[16-carbamoyl-31-carbamoylmethyl-10-(2-carboxyet...)
Affinity DataIC50:  1.50E+4nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230486(5-[(1Z)-({[(3R,5S)-5-{[(1S)-1-{[(1S)-1-carbamoyl-3...)
Affinity DataIC50:  1.60E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230467((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.60E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230463((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.60E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230455((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.60E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSHC-transforming protein 1(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50276397(4-((S)-2-acetamido-3-((S)-5-amino-1-((2-((S)-1-ami...)
Affinity DataIC50:  1.60E+4nMAssay Description:Displacement of FITC-tagged NH-(CH2)4-CO-phospho-tyrosine-glutamine-glycine-leucine-serine-amide from Shc Src homology 2 domain (unknown origin) by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSHC-transforming protein 1(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50276398(4-((S)-2-acetamido-3-((S)-5-amino-1-((2-((S)-1-ami...)
Affinity DataIC50:  1.70E+4nMAssay Description:Displacement of FITC-tagged NH-(CH2)4-CO-phospho-tyrosine-glutamine-glycine-leucine-serine-amide from Shc Src homology 2 domain (unknown origin) by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSHC-transforming protein 1(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50276391(4-((S)-2-acetamido-3-((S)-5-amino-1-((2-((S)-1-ami...)
Affinity DataIC50:  1.70E+4nMAssay Description:Displacement of FITC-tagged NH-(CH2)4-CO-phospho-tyrosine-glutamine-glycine-leucine-serine-amide from Shc Src homology 2 domain (unknown origin) by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230447((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.70E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230481((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.70E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230445((4S)-4-{[(1S)-1-carbamoyl-3-carboxypropyl]carbamoy...)
Affinity DataIC50:  1.80E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTumor susceptibility gene 101 protein(Homo sapiens (Human))
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50230454((4S)-4-{[(2S,3S)-3-{[(Z)-{[4-(benzyloxy)phenyl]met...)
Affinity DataIC50:  1.80E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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