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Found 65 with Last Name = 'fujieda' and Initial = 'h'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50468576(CHEMBL4281494)
Affinity DataIC50: <300nMAssay Description:Inhibition of [3H]-dofetilide binding to human ERG expressed in HEK293 cell membranes after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50468577(CHEMBL4283796)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human ERG expressed in HEK293 cells at -80 holding potential by whole patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213768(3-(4-(2-((4-(trifluoromethyl)benzyl)(benzo[d]thiaz...)
Affinity DataEC50:  4.46E+3nMAssay Description:Agonist activity at human PPARalpha receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213769(3-(4-(2-(benzo[d]thiazol-2-yl(thiophen-2-ylmethyl)...)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213768(3-(4-(2-((4-(trifluoromethyl)benzyl)(benzo[d]thiaz...)
Affinity DataEC50:  3.69E+3nMAssay Description:Agonist activity at human PPARgamma receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213771(3-(4-(2-((4-tert-butylbenzyl)(benzo[d]thiazol-2-yl...)
Affinity DataEC50:  6.34E+3nMAssay Description:Agonist activity at human PPARgamma receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213770(3-(4-(2-(benzyl(6-chlorobenzo[d]thiazol-2-yl)amino...)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213772(3-(4-(2-(benzo[d]thiazol-2-yl(benzyl)amino)ethoxy)...)
Affinity DataEC50:  1.17E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213773(3-(4-(2-(benzo[d]thiazol-2-yl(benzyl)amino)ethoxy)...)
Affinity DataEC50:  2.81E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213774(3-(4-(3-((6-chlorobenzo[d]thiazol-2-yl)(thiophen-2...)
Affinity DataEC50:  390nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213775(3-(4-(3-(benzo[d]thiazol-2-yl(benzyl)amino)propoxy...)
Affinity DataEC50:  2.55E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213771(3-(4-(2-((4-tert-butylbenzyl)(benzo[d]thiazol-2-yl...)
Affinity DataEC50:  4.88E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213777(3-(4-(2-(benzo[d]thiazol-2-yl(benzyl)amino)ethoxy)...)
Affinity DataEC50:  2.97E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213776(3-(4-(2-(benzyl(6-methylbenzo[d]thiazol-2-yl)amino...)
Affinity DataEC50:  2.61E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213768(3-(4-(2-((4-(trifluoromethyl)benzyl)(benzo[d]thiaz...)
Affinity DataEC50:  940nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50240347((9,12,15)-linolenic acid | (9Z,12Z,15Z)-octadeca-9...)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at human GPR120-Galpha16 fusion protein expressed in Flp-in HEK293 cells assessed as effect on intracellular calcium concentration b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50275055(4-{4-[2-(Phenyl-2-pyridinylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human GPR120-Galpha16 fusion protein expressed in Flp-in HEK293 cells assessed as effect on intracellular calcium concentration b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50275055(4-{4-[2-(Phenyl-2-pyridinylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  1.90E+4nMAssay Description:Agonist activity at human GPR40 expressed in T-REx HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50275158(4-{4-[2-(phenyl-2-thiazolylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  2.10E+4nMAssay Description:Agonist activity at human GPR40 expressed in T-REx HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50275158(4-{4-[2-(phenyl-2-thiazolylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GPR120-Galpha16 fusion protein expressed in Flp-in HEK293 cells assessed as effect on intracellular calcium concentration b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50240347((9,12,15)-linolenic acid | (9Z,12Z,15Z)-octadeca-9...)
Affinity DataEC50:  5.20E+3nMAssay Description:Agonist activity at human GPR40 expressed in T-REx HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387888(CHEMBL2058398)
Affinity DataEC50:  86nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Mus musculus)
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387889(CHEMBL2058666)
Affinity DataEC50:  159nMAssay Description:Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387890(CHEMBL2058388)
Affinity DataEC50:  2.61E+3nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387891(CHEMBL2058389)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387892(CHEMBL2058390)
Affinity DataEC50:  145nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387893(CHEMBL2058391)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387894(CHEMBL2058394)
Affinity DataEC50:  736nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387895(CHEMBL2058395)
Affinity DataEC50:  254nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387896(CHEMBL2058396)
Affinity DataEC50:  511nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387897(CHEMBL2058397)
Affinity DataEC50:  268nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387898(CHEMBL2058399)
Affinity DataEC50:  770nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387899(CHEMBL2058400)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387902(CHEMBL2058403)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387903(CHEMBL2058404)
Affinity DataEC50:  88nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387904(CHEMBL2058405)
Affinity DataEC50:  272nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387905(CHEMBL2058406)
Affinity DataEC50:  734nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387889(CHEMBL2058666)
Affinity DataEC50:  117nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387906(CHEMBL2058667)
Affinity DataEC50:  115nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387907(CHEMBL2058668)
Affinity DataEC50:  149nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387908(CHEMBL2058669)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387909(CHEMBL2058670)
Affinity DataEC50:  161nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387910(CHEMBL2058671)
Affinity DataEC50:  704nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387911(CHEMBL2058672)
Affinity DataEC50:  121nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387912(CHEMBL2058673)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387913(CHEMBL2058674)
Affinity DataEC50:  58nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Mus musculus)
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387893(CHEMBL2058391)
Affinity DataEC50:  224nMAssay Description:Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Mus musculus)
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387895(CHEMBL2058395)
Affinity DataEC50:  266nMAssay Description:Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Mus musculus)
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50387897(CHEMBL2058397)
Affinity DataEC50:  331nMAssay Description:Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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