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Found 54 with Last Name = 'fujii' and Initial = 'a'
TargetGlucagon receptor(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50122102(3-Cyano-4-hydroxy-benzoic acid [1-(2,3,5,6-tetrame...)
Affinity DataIC50:  2.30nMAssay Description:Antagonist activity against human glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in rat hepatocytes after 15 mins by cAMP dynamic2 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116666(4-Methyl-3,6-dihydro-1H-pyridin-(2Z)-ylideneamine ...)
Affinity DataIC50:  22nMAssay Description:The concentration required for inhibition of Inducible nitric oxide synthase in mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116674(6-Allyl-4-methyl-5,6-dihydro-1H-pyridin-(2Z)-ylide...)
Affinity DataIC50:  25nMAssay Description:The concentration required for inhibition of Inducible nitric oxide synthase in mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116674(6-Allyl-4-methyl-5,6-dihydro-1H-pyridin-(2Z)-ylide...)
Affinity DataIC50:  50nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116668(4-Methyl-6-propyl-5,6-dihydro-1H-pyridin-(2Z)-ylid...)
Affinity DataIC50:  60nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057824(CHEMBL3326175)
Affinity DataIC50:  87nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116668(4-Methyl-6-propyl-5,6-dihydro-1H-pyridin-(2Z)-ylid...)
Affinity DataIC50:  100nMAssay Description:The concentration required for inhibition of Inducible nitric oxide synthase in mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116667(4,5,5-Trimethyl-5,6-dihydro-1H-pyridin-(2Z)-yliden...)
Affinity DataIC50:  100nMAssay Description:The concentration required for inhibition of Inducible nitric oxide synthase in mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057820(CHEMBL3326174)
Affinity DataIC50:  160nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116670((4aR,7aR)-4-Methyl-1,4a,5,6,7,7a-hexahydro-[1]pyri...)
Affinity DataIC50:  170nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116676(4,6-Dimethyl-5,6-dihydro-1H-pyridin-(2Z)-ylideneam...)
Affinity DataIC50:  180nMAssay Description:Concentration required to inhibit Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116666(4-Methyl-3,6-dihydro-1H-pyridin-(2Z)-ylideneamine ...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116666(4-Methyl-3,6-dihydro-1H-pyridin-(2Z)-ylideneamine ...)
Affinity DataIC50:  230nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116676(4,6-Dimethyl-5,6-dihydro-1H-pyridin-(2Z)-ylideneam...)
Affinity DataIC50:  240nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057813(CHEMBL3326173)
Affinity DataIC50:  270nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50:  292nMAssay Description:Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in human hepatocytes after 15 mins by cAMP dynamic2 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116673(3,4-Dimethyl-5,6-dihydro-1H-pyridin-(2Z)-ylideneam...)
Affinity DataIC50:  310nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116673(3,4-Dimethyl-5,6-dihydro-1H-pyridin-(2Z)-ylideneam...)
Affinity DataIC50:  320nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116674(6-Allyl-4-methyl-5,6-dihydro-1H-pyridin-(2Z)-ylide...)
Affinity DataIC50:  360nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116667(4,5,5-Trimethyl-5,6-dihydro-1H-pyridin-(2Z)-yliden...)
Affinity DataIC50:  420nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057806(CHEMBL3326172)
Affinity DataIC50:  430nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116666(4-Methyl-3,6-dihydro-1H-pyridin-(2Z)-ylideneamine ...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116670((4aR,7aR)-4-Methyl-1,4a,5,6,7,7a-hexahydro-[1]pyri...)
Affinity DataIC50:  510nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116675(4,5-Dimethyl-5,6-dihydro-1H-pyridin-(2Z)-ylideneam...)
Affinity DataIC50:  510nMAssay Description:Concentration required to inhibit Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116675(4,5-Dimethyl-5,6-dihydro-1H-pyridin-(2Z)-ylideneam...)
Affinity DataIC50:  520nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116668(4-Methyl-6-propyl-5,6-dihydro-1H-pyridin-(2Z)-ylid...)
Affinity DataIC50:  580nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116666(4-Methyl-3,6-dihydro-1H-pyridin-(2Z)-ylideneamine ...)
Affinity DataIC50:  700nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057798(CHEMBL3326170)
Affinity DataIC50:  970nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of GLP-1R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50237936(4-Ethyl-5,6-dihydro-1H-pyridin-(2Z)-ylideneamine |...)
Affinity DataIC50:  1.20E+3nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116677((4aR,8aR)-4-Methyl-4a,5,6,7,8,8a-hexahydro-1H-quin...)
Affinity DataIC50:  1.40E+3nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057800(CHEMBL3326171)
Affinity DataIC50:  1.40E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50237936(4-Ethyl-5,6-dihydro-1H-pyridin-(2Z)-ylideneamine |...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116667(4,5,5-Trimethyl-5,6-dihydro-1H-pyridin-(2Z)-yliden...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116669(5,5-Dimethyl-5,6-dihydro-1H-pyridin-(2Z)-ylideneam...)
Affinity DataIC50:  2.80E+3nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057864(CHEMBL3325456)
Affinity DataIC50:  2.90E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057817(CHEMBL3326187)
Affinity DataIC50:  5.50E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116677((4aR,8aR)-4-Methyl-4a,5,6,7,8,8a-hexahydro-1H-quin...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057797(CHEMBL3326165)
Affinity DataIC50:  9.50E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057825(CHEMBL3326176)
Affinity DataIC50:  9.50E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50:  9.60E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057831(CHEMBL3326177)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50058003(CHEMBL3326186)
Affinity DataIC50:  2.40E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057859(CHEMBL3326181)
Affinity DataIC50:  2.70E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute

Curated by ChEMBL
LigandPNGBDBM50116669(5,5-Dimethyl-5,6-dihydro-1H-pyridin-(2Z)-ylideneam...)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057863(CHEMBL3326185)
Affinity DataIC50:  4.40E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057861(CHEMBL3326183)
Affinity DataIC50:  6.90E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057834(CHEMBL3326178)
Affinity DataIC50:  8.90E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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