Affinity DataIC50: 2.30nMAssay Description:Antagonist activity against human glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in rat hepatocytes after 15 mins by cAMP dynamic2 assayMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:The concentration required for inhibition of Inducible nitric oxide synthase in mouseMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:The concentration required for inhibition of Inducible nitric oxide synthase in mouseMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:The concentration required for inhibition of Inducible nitric oxide synthase in mouseMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:The concentration required for inhibition of Inducible nitric oxide synthase in mouseMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Concentration required to inhibit Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 292nMAssay Description:Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in human hepatocytes after 15 mins by cAMP dynamic2 assayMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Concentration required to inhibit Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 970nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of GLP-1R (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Concentration required to inhibit human Inducible nitric oxide synthase over expressed in A549 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 9.60E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Fukui Research Institute
Curated by ChEMBL
Fukui Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of human endothelial Nitric Oxide Synthase expressed in Sf-21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair