TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 5.60nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.40nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.90nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.70nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.70nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.20nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.80nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.90nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 9.10nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 9.5nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 10.7nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 10.8nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 10.8nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 640nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 730nMAssay Description:Antagonist activity at human vasopressin V1a expressed in AVP-stimulated HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair