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Found 20 with Last Name = 'gehrke' and Initial = 'l'
TargetTubulin beta-2B chain(Bos taurus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataKi:  180nMAssay Description:Binding constant at colchicine site of bovine brain tubulinMore data for this Ligand-Target Pair
TargetTubulin beta-2B chain(Bos taurus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50109343(1-Methyl-5-[(S)-5-(3,4,5-trimethoxy-phenyl)-4,5-di...)
Affinity DataKi:  630nMAssay Description:Binding constant at colchicine site of bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataKi:  780nMAssay Description:Binding constant at colchicine site of bovine brain tubulinMore data for this Ligand-Target Pair
TargetTubulin beta-2B chain(Bos taurus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50109342(1-Methyl-5-[(R)-5-(3,4,5-trimethoxy-phenyl)-4,5-di...)
Affinity DataKi:  3.69E+3nMAssay Description:Binding constant at colchicine site of bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding constant at colchicine site of bovine brain tubulinMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  1.20E+3nMAssay Description:Concentration required to inhibit polymerization of tubulinMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50006677(1,2,3-Trimethoxy-5-[(Z)-2-(4-methoxy-phenyl)-vinyl...)
Affinity DataIC50:  1.30E+3nMAssay Description:Concentration required to inhibit polymerization of tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50098052(3,4,5-Trimethoxy-benzenesulfonic acid 1-methyl-1H-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Concentration required to inhibit polymerization of tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50009565(CHEMBL312992 | Dimethyl-{4-[(Z)-2-(3,4,5-trimethox...)
Affinity DataIC50:  1.70E+3nMAssay Description:Concentration required to inhibit polymerization of tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50101086(CHEMBL20684 | E-7010 | N-(2-(4-hydroxyphenylamino)...)
Affinity DataIC50:  3.10E+3nMAssay Description:Concentration inhibiting tubulin polymerizationMore data for this Ligand-Target Pair
TargetTubulin beta-2B chain(Bos taurus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50109351(1-[5-(4-Amino-3-methyl-phenyl)-2-(3,4,5-trimethoxy...)
Affinity DataIC50:  3.40E+3nMAssay Description:Activity towards binding at colchicine site of bovine brain tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50101087(4-Methoxy-benzenesulfonic acid 2-((E)-2-pyridin-4-...)
Affinity DataIC50:  3.46E+3nMAssay Description:Concentration inhibiting tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50101098(4-Methoxy-benzenesulfonic acid 2-[(pyridine-4-carb...)
Affinity DataIC50:  3.73E+3nMAssay Description:Concentration inhibiting tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50101093(4-Methoxy-benzenesulfonic acid 2-[(pyridine-2-carb...)
Affinity DataIC50:  4.06E+3nMAssay Description:Concentration inhibiting tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50101085(4-Methoxy-benzenesulfonic acid 2-[(pyrazine-2-carb...)
Affinity DataIC50:  5.20E+3nMAssay Description:Concentration inhibiting tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50098051(3,4,5-Trimethoxy-benzenesulfonic acid 1H-indol-5-y...)
Affinity DataIC50:  6.60E+3nMAssay Description:Concentration required to inhibit polymerization of tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50098053(3-Amino-4-methoxy-benzenesulfonic acid 3,4,5-trime...)
Affinity DataIC50:  6.70E+3nMAssay Description:Concentration required to inhibit polymerization of tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50098050(4-Methoxy-benzenesulfonic acid 3,4,5-trimethoxy-ph...)
Affinity DataIC50:  8.20E+3nMAssay Description:Concentration required to inhibit polymerization of tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50098049(4-Dimethylamino-benzenesulfonic acid 3,4,5-trimeth...)
Affinity DataIC50:  1.60E+4nMAssay Description:Concentration required to inhibit polymerization of tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50098057(CHEMBL169800 | Toluene-4-sulfonic acid 3,4,5-trime...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit polymerization of tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed