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Found 11 with Last Name = 'gerasimov' and Initial = 'm'
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50081707(3-((R)-1-Methyl-pyrrolidin-2-ylmethyl)-1H-indol-6-...)
Affinity DataKi:  210nMAssay Description:Compound was tested for binding affinity using [3H]-MDL-100,907 at 5-hydroxytryptamine 2A receptor sites in rat cortical homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50081701(3-[2-(dimethylamino)ethyl]-1H-indol-4-ol | 4-hydro...)
Affinity DataKi:  390nMAssay Description:Compound was tested for binding affinity using [3H]-MDL-100,907 at 5-hydroxytryptamine 2A receptor sites in rat cortical homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50081704(5-Methoxy-3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1...)
Affinity DataKi:  400nMAssay Description:Compound was tested for binding affinity using [3H]-MDL-100,907 at 5-hydroxytryptamine 2A receptor sites in rat cortical homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50081705(3-(1-Methyl-pyrrolidin-3-yl)-1H-indol-4-ol | CHEMB...)
Affinity DataKi:  440nMAssay Description:Compound was tested for binding affinity using [3H]-MDL-100,907 at 5-hydroxytryptamine 2A receptor sites in rat cortical homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50081706(5-Methoxy-3-(1-methyl-pyrrolidin-3-yl)-1H-indole |...)
Affinity DataKi:  1.30E+3nMAssay Description:Compound was tested for binding affinity using [3H]-MDL-100,907 at 5-hydroxytryptamine 2A receptor sites in rat cortical homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM30707(2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)
Affinity DataKi:  1.60E+3nMAssay Description:Compound was tested for binding affinity using [3H]-MDL-100,907 at 5-hydroxytryptamine 2A receptor sites in rat cortical homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50081703(3-((S)-1-Methyl-pyrrolidin-2-ylmethyl)-1H-indol-6-...)
Affinity DataKi:  4.70E+3nMAssay Description:Compound was tested for binding affinity using [3H]-MDL-100,907 at 5-hydroxytryptamine 2A receptor sites in rat cortical homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50081702(5-Methoxy-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1...)
Affinity DataKi: >9.40E+3nMAssay Description:Compound was tested for binding affinity using [3H]-MDL-100,907 at 5-hydroxytryptamine 2A receptor sites in rat cortical homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Rattus norvegicus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50401019(CHEMBL2203661)
Affinity DataKi:  3.10E+4nMAssay Description:Inactivation of GABA-AT in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50118886(4-Amino-hex-5-enoic acid | CHEMBL89598 | US1018980...)
Affinity DataKi:  3.20E+6nMAssay Description:Inactivation of GABA-ATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target4-aminobutyrate aminotransferase, mitochondrial(Rattus norvegicus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50118886(4-Amino-hex-5-enoic acid | CHEMBL89598 | US1018980...)
Affinity DataKi:  1.00E+7nMAssay Description:Inactivation of GABA-AT in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed