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Found 365 with Last Name = 'graham' and Initial = 'dw'
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)
Affinity DataKi:  6.10nMAssay Description:Compound was tested for it''s ability to inhibit [3H]C18-PAF binding to PMN membrane receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023962(2-[(2,2-Dibromo-cyclopropanecarbonyl)-amino]-hex-2...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023979(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-7-(3...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024024(2-[(2,2-Dibromo-cyclopropanecarbonyl)-amino]-but-2...)
Affinity DataKi:  30nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023951(2-{6-Carboxy-6-[(2,2-dimethyl-cyclopropanecarbonyl...)
Affinity DataKi:  40nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024072(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-8-et...)
Affinity DataKi:  44nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023999(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hept...)
Affinity DataKi:  48nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024019(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-oct-...)
Affinity DataKi:  58nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)
Affinity DataKi:  59nMAssay Description:Compound was tested for it''s ability to inhibit [3H]C18-PAF binding to human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024071(2-[(2,2-Dichloro-cyclopropanecarbonyl)-amino]-oct-...)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367508(CHEMBL1907817)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367506(CHEMBL1907823)
Affinity DataKi:  80nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023983(2-[(2,2-Dichloro-cyclopropanecarbonyl)-amino]-but-...)
Affinity DataKi:  80nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023933(8-Cyano-2-[(2,2-dimethyl-cyclopropanecarbonyl)-ami...)
Affinity DataKi:  82nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024023(CHEMBL276215 | Sodium; 6-carboxy-6-[(2,2-dimethyl-...)
Affinity DataKi:  87nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024055(2-{6-Carboxy-6-[(2,2-dimethyl-cyclopropanecarbonyl...)
Affinity DataKi:  90nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023947(2,11-Bis-[(2,2-dimethyl-cyclopropanecarbonyl)-amin...)
Affinity DataKi:  92nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024044(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-dec-...)
Affinity DataKi:  96nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023992(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-7-ph...)
Affinity DataKi:  100nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50366241(CHEMBL297624 | L-652731)
Affinity DataKi:  103nMAssay Description:Inhibitory concentration required to inhibit PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023990(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hept...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023942(10-Bromo-2-[(2,2-dimethyl-cyclopropanecarbonyl)-am...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367502(CILASTATIN)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023995(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-dode...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024042(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-unde...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024045(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hex-...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)
Affinity DataKi:  116nMAssay Description:Compound was tested for it''s ability to inhibit [3H]C18-PAF binding to human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)
Affinity DataKi:  116nMAssay Description:Compound was tested for it''s ability to inhibit [3H]C18-PAF binding to human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024036(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-5-me...)
Affinity DataKi:  120nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024069(7-Carboxymethylsulfanyl-2-[(2,2-dimethyl-cycloprop...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024003(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-6-(3...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023971(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hex-...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024078(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-trid...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024059(7-Bromo-2-[(2,2-dimethyl-cyclopropanecarbonyl)-ami...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024012(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-8-me...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367507(CHEMBL1237318)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367505(CHEMBL1907816)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023963(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-6-me...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023946(4-Cyclohexyl-2-[(2,2-dimethyl-cyclopropanecarbonyl...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024053(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-7-me...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367509(CHEMBL1907822)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024005(9-Bromo-2-[(2,2-dimethyl-cyclopropanecarbonyl)-ami...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024066(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-non-...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024058(7-(2-Carboxy-2-oxo-ethylsulfanyl)-2-[(2,2-dimethyl...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023976((R)-2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-...)
Affinity DataKi:  170nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023972(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-8-me...)
Affinity DataKi:  170nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023980(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-8-me...)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50024008(CHEMBL11674 | {7-Carboxy-7-[(2,2-dichloro-cyclopro...)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50367503(CHEMBL1907818)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50023997(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-pent...)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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