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Found 167 with Last Name = 'green' and Initial = 'rc'
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041291(2-[(R)-3-(1,1-Dimethyl-2-phenyl-ethyl)-2,4,8-triox...)
Affinity DataKi:  0.930nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037348(1N-(3,3,3-trifluoro-1-isopropyl-2-oxopropyl)-2-(3-...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301315(CHEMBL568467 | N-(3,4-dimethyl-5-(morpholinomethyl...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377711(CHEMBL256962)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277153(4-methyl-3-(morpholinosulfonyl)-N-((1S,2R,4R)-1,3,...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377707(CHEMBL255474)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50036127(CHEMBL11391 | {2-Oxo-6-phenyl-1-[(3,3,3-trifluoro-...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377706(CHEMBL256110)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037341(4-{2-Oxo-6-phenyl-1-[(3,3,3-trifluoro-1-isopropyl-...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377705(CHEMBL442447)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50036112(CHEMBL11403 | {6-Oxo-2-phenyl-1-[(3,3,3-trifluoro-...)
Affinity DataKi:  6.60nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037375(CHEMBL275043 | {2-Oxo-6-phenyl-1-[(3,3,3-trifluoro...)
Affinity DataKi:  8nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377704(CHEMBL255096)
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50036103(CHEMBL11098 | {2-(4-Fluoro-phenyl)-6-oxo-1-[(3,3,3...)
Affinity DataKi:  8.20nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301316(CHEMBL568468 | N-(3,4-dimethyl-5-(morpholinomethyl...)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377710(CHEMBL256753)
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377703(CHEMBL258243)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377709(CHEMBL256754)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037100(2,2-Dimethyl-propionic acid 3-{5-benzyloxycarbonyl...)
Affinity DataKi:  12nMAssay Description:The compound was tested in vitro for ability to inhibit human leukocyte elastase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50036078(1-Oxo-3-phenyl-2-[(3,3,3-trifluoro-1-isopropyl-2-o...)
Affinity DataKi:  13nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377708(CHEMBL256752)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301312(3,3-difluoro-2-methyl-N-(4-methyl-3-(morpholinomet...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301306(2-methyl-N-(4-methyl-3-(morpholinomethyl)-5-(trifl...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037342(1N-(3,3,3-trifluoro-1-isopropyl-2-oxopropyl)-2-(3-...)
Affinity DataKi:  18nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301317(4-methyl-3-(morpholinomethyl)-N-((1S,4R)-1,3,3-tri...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377702(CHEMBL258244)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037117(2,2-Dimethyl-propionic acid 4-{5-benzyloxycarbonyl...)
Affinity DataKi:  32nMAssay Description:The compound was tested in vitro for ability to inhibit human leukocyte elastase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377706(CHEMBL256110)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037111(CHEMBL104303 | {5-(4-Hydroxy-benzyl)-2-oxo-1-[(3,3...)
Affinity DataKi:  34nMAssay Description:The compound was tested in vitro for ability to inhibit human leukocyte elastase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037102(CHEMBL75936 | {2-Oxo-5-[3-(2,2,2-trifluoro-acetyla...)
Affinity DataKi:  36nMAssay Description:The compound was tested in vitro for ability to inhibit human leukocyte elastase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301307(CHEMBL577487 | N-(2-fluoro-4-methyl-5-(morpholinom...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50036122(CHEMBL11336 | {2-(4-Fluoro-phenyl)-6-oxo-1-[(3,3,3...)
Affinity DataKi:  40nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037110(CHEMBL107291 | {5-Benzyl-2-oxo-1-[(3,3,3-trifluoro...)
Affinity DataKi:  40nMAssay Description:The compound was tested in vitro for ability to inhibit human leukocyte elastase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037105(Acetic acid 3-{5-benzyloxycarbonylamino-6-oxo-1-[(...)
Affinity DataKi:  42nMAssay Description:The compound was tested in vitro for ability to inhibit human leukocyte elastase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301318(4-methyl-3-(2-morpholinoethyl)-N-((1S,4R)-1,3,3-tr...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037113(CHEMBL104289 | [2-Oxo-1-[(3,3,3-trifluoro-1-isopro...)
Affinity DataKi:  47nMAssay Description:The compound was tested in vitro for ability to inhibit human leukocyte elastase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377701(CHEMBL404650)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037116(CHEMBL107966 | N-{5-Benzyl-2-oxo-1-[(3,3,3-trifluo...)
Affinity DataKi:  48nMAssay Description:The compound was tested in vitro for ability to inhibit human leukocyte elastase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377704(CHEMBL255096)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037098(CHEMBL104032 | N-{5-Benzyl-2-oxo-1-[(3,3,3-trifluo...)
Affinity DataKi:  51nMAssay Description:The compound was tested in vitro for ability to inhibit human leukocyte elastase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50036127(CHEMBL11391 | {2-Oxo-6-phenyl-1-[(3,3,3-trifluoro-...)
Affinity DataKi:  55nMAssay Description:The compound was evaluated for the binding affinity against bovine pancreatic chymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301319(4-methyl-3-(3-morpholinopropyl)-N-((1S,4R)-1,3,3-t...)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037118(CHEMBL106793 | N-{5-Benzyl-2-oxo-1-[(3,3,3-trifluo...)
Affinity DataKi:  70nMAssay Description:The compound was tested in vitro for ability to inhibit human leukocyte elastase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301313(2-methyl-N-(4-methyl-3-(morpholinomethyl)phenyl)cy...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50037099(CHEMBL104557 | {5-(4-Fluoro-benzyl)-2-oxo-1-[(3,3,...)
Affinity DataKi:  71nMAssay Description:The compound was tested in vitro for ability to inhibit human leukocyte elastase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50377705(CHEMBL442447)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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