TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of Rolipram binding to Phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Tested for inhibitory activity against Coagulation factor XaMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 97nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Sw 8 Rh£Ne-Poulenc Rorer Central Research
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Binding affinity at Phosphodiesterase 4 by measuring displacement of (+/-)-[3H]- Rolipram to guinea pig brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 620nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 620nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: >1.20E+3nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: >1.20E+3nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: >1.20E+3nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: >1.20E+3nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: >1.20E+3nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: >1.20E+3nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: >1.20E+3nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: >1.20E+3nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair