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Found 44 with Last Name = 'hasegawa' and Initial = 'h'
TargetProstaglandin-H2 D-isomerase(Homo sapiens (Human))
Shionogi

Curated by PDSP Ki Database
LigandPNGBDBM50008805(7-(3-Benzenesulfonylamino-bicyclo[2.2.1]hept-2-yl)...)
Affinity DataKi:  0.340nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin-H2 D-isomerase(GUINEA PIG)
Shionogi

Curated by PDSP Ki Database
LigandPNGBDBM50008805(7-(3-Benzenesulfonylamino-bicyclo[2.2.1]hept-2-yl)...)
Affinity DataKi:  0.490nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin-H2 D-isomerase(Homo sapiens (Human))
Shionogi

Curated by PDSP Ki Database
LigandPNGBDBM50060462((Z)-7-{(1R,2R,3S,5S)-2-[(5-Hydroxy-benzo[b]thiophe...)
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin-H2 D-isomerase(Homo sapiens (Human))
Shionogi

Curated by PDSP Ki Database
LigandPNGBDBM50060462((Z)-7-{(1R,2R,3S,5S)-2-[(5-Hydroxy-benzo[b]thiophe...)
Affinity DataKi:  24.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin-H2 D-isomerase(GUINEA PIG)
Shionogi

Curated by PDSP Ki Database
LigandPNGBDBM50060462((Z)-7-{(1R,2R,3S,5S)-2-[(5-Hydroxy-benzo[b]thiophe...)
Affinity DataKi:  193nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin-H2 D-isomerase(Homo sapiens (Human))
Shionogi

Curated by PDSP Ki Database
LigandPNGBDBM85347(BWA868C | CAS_122021 | NSC_122021)
Affinity DataKi:  2.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin-H2 D-isomerase(Homo sapiens (Human))
Shionogi

Curated by PDSP Ki Database
LigandPNGBDBM50008805(7-(3-Benzenesulfonylamino-bicyclo[2.2.1]hept-2-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEndothelin-converting enzyme 1(Rattus norvegicus (Rat))
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50112397(CHEMBL22323 | Sodium;4-chloro-N-{[(4-cyano-3-methy...)
Affinity DataIC50:  42nMAssay Description:Tested in vitro for inhibition of Endothelin-converting enzyme (ECE) of rat lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Rattus norvegicus (Rat))
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50040413((S)-2-{(S)-2-[Hydroxy-(3,4,5-trihydroxy-6-methyl-t...)
Affinity DataIC50:  690nMAssay Description:Tested in vitro for inhibition of Endothelin-converting enzyme (ECE) of rat lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Rattus norvegicus (Rat))
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50112394(5-{(2Z)-2-[[(E)-(4-propylphenyl)diazenyl](phenyl)m...)
Affinity DataIC50:  2.60E+3nMAssay Description:Tested in vitro for inhibition of Endothelin-converting enzyme (ECE) of rat lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Rattus norvegicus (Rat))
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50112393(5-{(2Z)-2-[[(E)-(4-secbutylphenyl)diazenyl](phenyl...)
Affinity DataIC50:  2.70E+3nMAssay Description:Tested in vitro for inhibition of Endothelin-converting enzyme (ECE) of rat lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Rattus norvegicus (Rat))
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50112401(5-{(2Z)-2-[[(E)-(4-isopropylphenyl)diazenyl](pheny...)
Affinity DataIC50:  3.40E+3nMAssay Description:Tested in vitro for inhibition of Endothelin-converting enzyme (ECE) of rat lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Rattus norvegicus (Rat))
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50112396(5-{(2Z)-2-[[(E)-(4-cyclohexylphenyl)diazenyl](phen...)
Affinity DataIC50:  3.60E+3nMAssay Description:Tested in vitro for inhibition of Endothelin-converting enzyme (ECE) of rat lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Rattus norvegicus (Rat))
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50112400(5-{(2Z)-2-[[(E)-(4-tertbutylphenyl)diazenyl](pheny...)
Affinity DataIC50:  3.80E+3nMAssay Description:Tested in vitro for inhibition of Endothelin-converting enzyme (ECE) of rat lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Rattus norvegicus (Rat))
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50112398(5-{(2Z)-2-[[(E)-(4-ethylphenyl)diazenyl](phenyl)me...)
Affinity DataIC50:  3.80E+3nMAssay Description:Tested in vitro for inhibition of Endothelin-converting enzyme (ECE) of rat lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Rattus norvegicus (Rat))
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50112395(5-{(2Z)-2-[[(E)-(4-methylphenyl)diazenyl](phenyl)m...)
Affinity DataIC50:  8.40E+3nMAssay Description:Tested in vitro for inhibition of Endothelin-converting enzyme (ECE) of rat lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Rattus norvegicus (Rat))
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50112399(1-phenyl-5-((2Z)-2-{phenyl[(E)-phenyldiazenyl]meth...)
Affinity DataIC50:  1.00E+4nMAssay Description:Tested in vitro for inhibition of Endothelin-converting enzyme (ECE) of rat lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179868(CHEMBL203454 | N-methyl-N-(4-(2,2,2-trifluoro-1-hy...)
Affinity DataEC50: >5.00E+3nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179869(CHEMBL203682 | N-methyl-N-[4-(2,2,2-trifluoro-1-hy...)
Affinity DataEC50:  200nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179865(2-cyano-N-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxyprop...)
Affinity DataEC50:  700nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179866(CHEMBL380851 | N-(4-(1,1,1,3,3,3-hexafluoro-2-hydr...)
Affinity DataEC50:  40nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)
Affinity DataEC50:  10nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179870(CHEMBL206445 | N1-(4-(1,1,1,3,3,3-hexafluoro-2-hyd...)
Affinity DataEC50:  80nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM20164((1S,2R,5S,10S,11S,14R,15R)-14-[(2R)-4-[(2S)-3,3-di...)
Affinity DataEC50:  500nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179871(CHEMBL383657 | N-methyl-N-(4-(1,1,1-trifluoro-2-hy...)
Affinity DataEC50:  5.00E+3nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179872(CHEMBL206674 | biphenyl-3-sulfonic acid methyl-[4-...)
Affinity DataEC50:  30nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179876(1,1,1,3,3,3-hexafluoro-2-(4-(phenylsulfonyl)-3,4-d...)
Affinity DataEC50:  100nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179877(1,1,1,3,3,3-hexafluoro-2-(1-(phenylsulfonyl)-1,2,3...)
Affinity DataEC50:  30nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179873(CHEMBL204282 | N-(3-(1,1,1,3,3,3-hexafluoro-2-hydr...)
Affinity DataEC50:  1.00E+3nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179878(CHEMBL206192 | N-(4-(1,1,1,3,3,3-hexafluoro-2-hydr...)
Affinity DataEC50:  600nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179874(CHEMBL380249 | N-(2-chloro-4-(1,1,1,3,3,3-hexafluo...)
Affinity DataEC50:  200nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179875(4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-N-...)
Affinity DataEC50:  100nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179879(4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-N-...)
Affinity DataEC50:  200nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179880(1,1,1,3,3,3-hexafluoro-2-(1-(phenylsulfonyl)indoli...)
Affinity DataEC50:  50nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179859(CHEMBL203606 | isobutyl 4-(1,1,1,3,3,3-hexafluoro-...)
Affinity DataEC50:  100nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179858(1,1,1,3,3,3-hexafluoro-2-(1-(phenylsulfonyl)-2,3,4...)
Affinity DataEC50:  10nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179857(4-cyano-N-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxyprop...)
Affinity DataEC50:  2.00E+3nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179856(CHEMBL205770 | N-(3-chloro-4-(1,1,1,3,3,3-hexafluo...)
Affinity DataEC50: >5.00E+3nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179867(CHEMBL382792 | N-(4-(1,1,1,3,3,3-hexafluoro-2-hydr...)
Affinity DataEC50:  4.00E+3nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179864(3-cyano-N-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxyprop...)
Affinity DataEC50:  20nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179863(CHEMBL379225 | N-(4-(1,1,1,3,3,3-hexafluoro-2-hydr...)
Affinity DataEC50:  100nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179860(CHEMBL206738 | N-cyclopentyl-N-(4-(1,1,1,3,3,3-hex...)
Affinity DataEC50:  8nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179861(CHEMBL380711 | N-(4-(1,1,1,3,3,3-hexafluoro-2-hydr...)
Affinity DataEC50:  3.00E+3nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50179862(CHEMBL203824 | N-(4-(1,1,1,3,3,3-hexafluoro-2-meth...)
Affinity DataEC50:  1.00E+3nMAssay Description:Activity against LXR alpha transiently transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed