Affinity DataKi: 1nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.2kJ/molepH: 7.2 T: 2°CAssay Description:The 11beta-HSD1 enzyme assay was carried out in the replica plates of the compounds in reaction buffer containing substrate mixture [3H]-cortisone/NA...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibitory activity against recombinant human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 12nM ΔG°: -44.8kJ/molepH: 7.2 T: 2°CAssay Description:The 11beta-HSD1 enzyme assay was carried out in the replica plates of the compounds in reaction buffer containing substrate mixture [3H]-cortisone/NA...More data for this Ligand-Target Pair
Affinity DataKi: 12.2nMAssay Description:Displacement of [3H]-cortisone human 17beta-HSD1 expressed in Escherichia coli after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.8nMAssay Description:Displacement of [3H]-cortisone human 17beta-HSD1 expressed in Escherichia coli after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nM ΔG°: -44.6kJ/molepH: 7.2 T: 2°CAssay Description:The 11beta-HSD1 enzyme assay was carried out in the replica plates of the compounds in reaction buffer containing substrate mixture [3H]-cortisone/NA...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 13nM ΔG°: -44.6kJ/molepH: 7.2 T: 2°CAssay Description:The 11beta-HSD1 enzyme assay was carried out in the replica plates of the compounds in reaction buffer containing substrate mixture [3H]-cortisone/NA...More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 14nM ΔG°: -44.4kJ/molepH: 7.2 T: 2°CAssay Description:The 11beta-HSD1 enzyme assay was carried out in the replica plates of the compounds in reaction buffer containing substrate mixture [3H]-cortisone/NA...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibitory activity against recombinant human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 17.3nMAssay Description:Displacement of [3H]-cortisone human 17beta-HSD1 expressed in Escherichia coli after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibitory activity against recombinant human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 20nM ΔG°: -43.5kJ/molepH: 7.2 T: 2°CAssay Description:The 11beta-HSD1 enzyme assay was carried out in the replica plates of the compounds in reaction buffer containing substrate mixture [3H]-cortisone/NA...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of human 11betaHSD1 by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair