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Found 39 with Last Name = 'kaczmarek' and Initial = 'r'
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50350515(CHEMBL1812067)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81576(AppppA analog, 6 (X=S))
Affinity DataKi:  35nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50350516(CHEMBL1812066)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50350514(CHEMBL1812068)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50350513(CHEMBL1812069)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50350512(CHEMBL1812070)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81584(AppppA analog, 12 (X=S))
Affinity DataKi:  40nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81586(AppppA analog, 13 (X=S))
Affinity DataKi:  65nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81590(AppppA analog, 15 (X=S))
Affinity DataKi:  78nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81593(AppppA analog, 17 (X=S))
Affinity DataKi:  110nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81575(AppppA analog, 5 (X=S))
Affinity DataKi:  220nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81580(AppppA analog, 9 (X=S))
Affinity DataKi:  230nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81592(AppppA analog, 17 (X=O))
Affinity DataKi:  420nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81588(AppppA analog, 14 (X=S))
Affinity DataKi:  700nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81587(AppppA analog, 14 (X=O))
Affinity DataKi:  900nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81583(AppppA analog, 12 (X=O))
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81574(AppppA analog, 5 (X=O))
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81589(AppppA analog, 15 (X=O))
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81570(AppppA analog, 1 (X=O))
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81571(AppppA analog, 2 (X=S))
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81591(AppppA analog, 16 (X=S))
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81579(AppppA analog, 8 (X=S))
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81585(AppppA analog, 13 (X=O))
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81581(AppppA analog, 10 (X=S))
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81577(AppppA analog, 6 (X=O))
Affinity DataKi:  4.70E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81582(AppppA analog, 11 (X=S))
Affinity DataKi:  5.20E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81578(AppppA analog, 7 (X=S))
Affinity DataKi:  7.60E+4nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81572(AppppA analog, 3 (X=S))
Affinity DataKi:  8.60E+4nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81573(AppppA analog, 4 (X=S))
Affinity DataKi:  8.60E+4nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50001207(CHEMBL3236423)
Affinity DataEC50: >5.00E+5nMAssay Description:Inhibition of human DNA polymerase alpha using dCTP as substrate assessed as single base extension reaction after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50001208(CHEMBL3236424)
Affinity DataEC50:  7.00E+4nMAssay Description:Inhibition of human DNA polymerase alpha using dCTP as substrate assessed as single base extension reaction after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50001209(CHEMBL3236425)
Affinity DataEC50:  4.10E+5nMAssay Description:Inhibition of human DNA polymerase alpha using dCTP as substrate assessed as single base extension reaction after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50001210(CHEMBL3236426)
Affinity DataEC50: >5.00E+5nMAssay Description:Inhibition of human DNA polymerase alpha using dCTP as substrate assessed as single base extension reaction after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50001206(CHEMBL3236422)
Affinity DataEC50:  2.50E+5nMAssay Description:Inhibition of human DNA polymerase alpha using dCTP as substrate assessed as single base extension reaction after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50001205(CHEMBL3236421)
Affinity DataEC50: >5.00E+5nMAssay Description:Inhibition of human DNA polymerase alpha using dCTP as substrate assessed as single base extension reaction after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50001204(CHEMBL3236420)
Affinity DataEC50: >5.00E+5nMAssay Description:Inhibition of human DNA polymerase alpha using dCTP as substrate assessed as single base extension reaction after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50001143(CHEMBL3236419)
Affinity DataEC50: >5.00E+5nMAssay Description:Inhibition of human DNA polymerase alpha using dCTP as substrate assessed as single base extension reaction after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50001141(CHEMBL3236417)
Affinity DataEC50:  3.50E+5nMAssay Description:Inhibition of human DNA polymerase alpha using dCTP as substrate assessed as single base extension reaction after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50001142(CHEMBL3236418)
Affinity DataEC50:  8.00E+4nMAssay Description:Inhibition of human DNA polymerase alpha using dCTP as substrate assessed as single base extension reaction after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed