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Found 327 with Last Name = 'katada' and Initial = 'j'
TargetChymotrypsinogen A(Bos taurus (bovine))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073123((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataKi:  4.5nMAssay Description:Compound was evaluated for inactivation of bovine alpha-Chymotrypsin Kinetic constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073127((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataKi:  70nMAssay Description:Compound was evaluated for inactivation of bovine alpha-Chymotrypsin Kinetic constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073126((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataKi:  340nMAssay Description:Compound was evaluated for inactivation of bovine alpha-Chymotrypsin Kinetic constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073125((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataKi:  1.20E+4nMAssay Description:Compound was evaluated for inactivation of bovine alpha-Chymotrypsin Kinetic constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073123((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataIC50:  0.700nMAssay Description:Compound was tested by chromogenic assay for the inhibition of serine proteases like Porcine ElastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073139(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-4-phenyl...)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory activity against human leukocyte cathepsin G (h-CG)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Bos taurus)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073123((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataIC50:  1.60nMAssay Description:In vitro inhibition of bovine alpha chymotrypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Bos taurus)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073123((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataIC50:  1.60nMAssay Description:In vitro inhibition of bovine alpha chymotrypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073139(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-4-phenyl...)
Affinity DataIC50:  2.10nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Bos taurus)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073139(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-4-phenyl...)
Affinity DataIC50:  2.10nMAssay Description:In vitro inhibition of bovine alpha chymotrypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064943((1-{3-[2-Fluoro-4-(imino-thiazolidin-3-yl-methyl)-...)
Affinity DataIC50:  2.30nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064930(CHEMBL77113 | {1-[3-(4-Carbamimidoyl-benzoylamino)...)
Affinity DataIC50:  2.60nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Bos taurus)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073123((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataIC50:  2.60nMAssay Description:In vitro inhibition of bovine alpha chymotrypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064941(CHEMBL78295 | {1-[3-(4-Carbamimidoyl-2-fluoro-benz...)
Affinity DataIC50:  2.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064942(CHEMBL74908 | {1-[3-(4-Carbamimidoyl-benzoylamino)...)
Affinity DataIC50:  2.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064935(CHEMBL312368 | {1-[3-(4-Carbamimidoyl-2-fluoro-ben...)
Affinity DataIC50:  2.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064922(CHEMBL432915 | {1-[3-(4-Carbamimidoyl-benzoylamino...)
Affinity DataIC50:  3.80nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064920((1-{3-[2-Fluoro-4-(imino-morpholin-4-yl-methyl)-be...)
Affinity DataIC50:  4nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064938(CHEMBL77635 | {1-[3-(4-Carbamimidoyl-2-fluoro-benz...)
Affinity DataIC50:  4.30nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064926(CHEMBL77404 | {1-[3-(4-Carbamimidoyl-benzoylamino)...)
Affinity DataIC50:  5nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075109(1,1-dimethyl-2-phenylcarboxamidoheptanoic anhydrid...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against human chymase (h-chymase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064921(CHEMBL75645 | {1-[3-(4-Carbamimidoyl-benzoylamino)...)
Affinity DataIC50:  5.10nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064927(CHEMBL76845 | {1-[3-(4-Carbamimidoyl-benzoylamino)...)
Affinity DataIC50:  5.30nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075109(1,1-dimethyl-2-phenylcarboxamidoheptanoic anhydrid...)
Affinity DataIC50:  5.30nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064928(CHEMBL78119 | [1-(3-{2-Fluoro-4-[imino-(4-methyl-p...)
Affinity DataIC50:  5.40nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064931(CHEMBL75623 | {1-[3-(2-Fluoro-4-{[4-(4-fluoro-phen...)
Affinity DataIC50:  5.60nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075107(1,1-dimethyl-4-phenyl-2-propylcarboxamidopentanoic...)
Affinity DataIC50:  5.60nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075107(1,1-dimethyl-4-phenyl-2-propylcarboxamidopentanoic...)
Affinity DataIC50:  5.60nMAssay Description:Inhibitory activity against human chymase (h-chymase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064917(CHEMBL74553 | {1-[3-(4-Carbamimidoyl-2-fluoro-benz...)
Affinity DataIC50:  5.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064918(CHEMBL76882 | [1-(3-{2-Fluoro-4-[(4-hydroxy-piperi...)
Affinity DataIC50:  5.80nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075109(1,1-dimethyl-2-phenylcarboxamidoheptanoic anhydrid...)
Affinity DataIC50:  6.40nMAssay Description:Inhibitory activity against human leukocyte cathepsin G (h-CG)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064939((1-{3-[2-Fluoro-4-(imino-pyrrolidin-1-yl-methyl)-b...)
Affinity DataIC50:  7nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073123((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataIC50:  8.40nMAssay Description:Compound was tested by chromogenic assay for the inhibition of serine proteases like Human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064934(CHEMBL76851 | {1-[3-(4-Carbamimidoyl-benzoylamino)...)
Affinity DataIC50:  8.60nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073123((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataIC50:  8.60nMAssay Description:Compound was tested by chromogenic assay for the inhibition of serine proteases like Porcine ElastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073123((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataIC50:  8.60nMAssay Description:Compound was tested by chromogenic assay for the inhibition of serine proteases like Porcine ElastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073123((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataIC50:  8.70nMAssay Description:Compound was tested by chromogenic assay for the inhibition of serine proteases like Human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073123((S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-nonan...)
Affinity DataIC50:  8.70nMAssay Description:Compound was tested by chromogenic assay for the inhibition of serine proteases like Human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075107(1,1-dimethyl-4-phenyl-2-propylcarboxamidopentanoic...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075107(1,1-dimethyl-4-phenyl-2-propylcarboxamidopentanoic...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064919(CHEMBL76960 | {1-[(E)-3-(4-Carbamimidoyl-benzoylam...)
Affinity DataIC50:  13nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075114(1,1-dimethyl-2-phenylcarboxamidooctanoic anhydride...)
Affinity DataIC50:  13nMAssay Description:Inhibitory activity against human chymase (h-chymase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075110(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-2-phenyl...)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity against human leukocyte cathepsin G (h-CG)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075110(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-2-phenyl...)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075106(1,1-dimethyl-4-phenyl-2-phenylcarboxamidopentanoic...)
Affinity DataIC50:  18nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075106(1,1-dimethyl-4-phenyl-2-phenylcarboxamidopentanoic...)
Affinity DataIC50:  18nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075106(1,1-dimethyl-4-phenyl-2-phenylcarboxamidopentanoic...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against human chymase (h-chymase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075106(1,1-dimethyl-4-phenyl-2-phenylcarboxamidopentanoic...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064932(CHEMBL76555 | {1-[3-(4-Carbamimidoyl-benzoylamino)...)
Affinity DataIC50:  21nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075107(1,1-dimethyl-4-phenyl-2-propylcarboxamidopentanoic...)
Affinity DataIC50:  21nMAssay Description:Inhibitory activity against human leukocyte cathepsin G (h-CG)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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