Affinity DataIC50: 140nMAssay Description:In vitro inhibitory concentration against Muscarinic acetylcholine receptor derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of smooth muscle cell ACAT activity for cells stimulated by cationized LDL.More data for this Ligand-Target Pair
Affinity DataIC50: 311nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 406nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 431nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 446nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 484nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 629nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 721nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 740nMAssay Description:Compound was evaluated for the effect on Cholesterol O-Acyltransferase (ACAT) in Liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 810nMAssay Description:Compound was evaluated for the effect on Cholesterol O-Acyltransferase (ACAT) in intestinal microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 952nMAssay Description:In vitro inhibitory concentration against ACAT derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 976nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+3nMAssay Description:In vitro inhibitory concentration against ACAT derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+3nMAssay Description:Compound was evaluated for the effect on Cholesterol O-Acyltransferase (ACAT) in Aorta (homogenate Low-density lipoproteins (LDL)More data for this Ligand-Target Pair
Affinity DataIC50: 1.31E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 1.44E+3nMAssay Description:In vitro inhibitory concentration against ACAT derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.71E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 1.83E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 2.24E+3nMAssay Description:In vitro inhibitory concentration against Muscarinic acetylcholine receptor derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.62E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 2.86E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.01E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 3.18E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.28E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.54E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.62E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 3.62E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.77E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 3.89E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.04E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.41E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.53E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 4.59E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.83E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.95E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.64E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.81E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.06E+3nMAssay Description:Inhibition of smooth muscle cell ACAT activity for cells stimulated by native LDL.More data for this Ligand-Target Pair
Affinity DataIC50: 6.30E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.85E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.55E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.69E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.49E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.19E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.54E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair