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Found 91 with Last Name = 'khalaf' and Initial = 'ai'
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206172(1-(benzo[d][1,3]dioxol-5-ylmethyl)-2,3,4,9-tetrahy...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206189(1-(2-(propylthio)benzyl)-2,3,4,9-tetrahydro-1H-pyr...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206163(1-(3-Methoxy-benzyl)-2,3,4,9-tetrahydro-1H-beta-ca...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206164(1-(2-(methylthio)benzyl)-2,3,4,9-tetrahydro-1H-pyr...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206169(1-(benzo[d][1,3]dioxol-5-ylmethyl)-6-methoxy-2,3,4...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206175(1-(3-methoxybenzyl)-6-methoxy-2,3,4,9-tetrahydro-1...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206186(2-fluoro-6-((2,3,4,9-tetrahydro-1H-pyrido[3,4-b]in...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206168(2,9-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibe...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206183((E)-6-((benzyl(methyl)amino)methyleneamino)-2,3-di...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206178((E)-6-((3,4-dihydroisoquinolin-2(1H)-yl)methylenea...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206161(1-(4-(methylthio)benzyl)-2,3,4,9-tetrahydro-1H-pyr...)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206174((E)-6-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206190((E)-3-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206173((E)-7-((3,4-dihydroisoquinolin-2(1H)-yl)methylenea...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206165((E)-7-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206162((E)-N-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206177((E)-3-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206192((E)-6-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206184((E)-N-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206162((E)-N-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206165((E)-7-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206192((E)-6-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206190((E)-3-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206184((E)-N-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206170(1-(3-methoxyphenyl)-4,9-dihydro-3H-pyrido[3,4-b]in...)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206177((E)-3-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206174((E)-6-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206182(3-(2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)p...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206173((E)-7-((3,4-dihydroisoquinolin-2(1H)-yl)methylenea...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206175(1-(3-methoxybenzyl)-6-methoxy-2,3,4,9-tetrahydro-1...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206163(1-(3-Methoxy-benzyl)-2,3,4,9-tetrahydro-1H-beta-ca...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206178((E)-6-((3,4-dihydroisoquinolin-2(1H)-yl)methylenea...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206183((E)-6-((benzyl(methyl)amino)methyleneamino)-2,3-di...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206178((E)-6-((3,4-dihydroisoquinolin-2(1H)-yl)methylenea...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206193(1-(3-methoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206177((E)-3-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206169(1-(benzo[d][1,3]dioxol-5-ylmethyl)-6-methoxy-2,3,4...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206180(9,10-dimethoxy-7-methyl-5,8,13,13a-tetrahydro-6H-[...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206187((E)-methyl 6-((6,7-dimethoxy-3,4-dihydroisoquinoli...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206176((E)-tert-butyl 6-((6,7-dimethoxy-3,4-dihydroisoqui...)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206173((E)-7-((3,4-dihydroisoquinolin-2(1H)-yl)methylenea...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206171((E)-6-((3,4-dihydroisoquinolin-2(1H)-yl)methylenea...)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206171((E)-6-((3,4-dihydroisoquinolin-2(1H)-yl)methylenea...)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206166((E)-3-(butylthio)-N-((6,7-dimethoxy-3,4-dihydroiso...)
Affinity DataKi:  3.10E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206188(6-methoxy-1-(3-methoxyphenyl)-4,9-dihydro-3H-pyrid...)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206167((E)-N-benzyl-N'-(3-hydroxy-2,3-dihydro-1H-inden-5-...)
Affinity DataKi:  3.60E+3nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206183((E)-6-((benzyl(methyl)amino)methyleneamino)-2,3-di...)
Affinity DataKi:  4.50E+3nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206166((E)-3-(butylthio)-N-((6,7-dimethoxy-3,4-dihydroiso...)
Affinity DataKi:  4.50E+3nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206172(1-(benzo[d][1,3]dioxol-5-ylmethyl)-2,3,4,9-tetrahy...)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206180(9,10-dimethoxy-7-methyl-5,8,13,13a-tetrahydro-6H-[...)
Affinity DataKi:  5.00E+3nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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