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Found 255 with Last Name = 'kim' and Initial = 'kb'
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50109593(2-Benzyl-3-mercapto-propionic acid | 2-Mercaptomet...)
Affinity DataKi:  11nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50109593(2-Benzyl-3-mercapto-propionic acid | 2-Mercaptomet...)
Affinity DataKi:  11nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279954(3-(3-Fluoro-phenyl)-2-mercaptomethyl-propionic aci...)
Affinity DataKi:  35nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279947(3-(4-Fluoro-phenyl)-2-mercaptomethyl-propionic aci...)
Affinity DataKi:  37nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279947(3-(4-Fluoro-phenyl)-2-mercaptomethyl-propionic aci...)
Affinity DataKi:  37nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279958(3-(2-Fluoro-phenyl)-2-mercaptomethyl-propionic aci...)
Affinity DataKi:  45nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279960(2-Mercaptomethyl-3-phenyl-butyric acid | CHEMBL109...)
Affinity DataKi:  105nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279955(2-Mercaptomethyl-3-p-tolyl-propionic acid | CHEMBL...)
Affinity DataKi:  112nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279955(2-Mercaptomethyl-3-p-tolyl-propionic acid | CHEMBL...)
Affinity DataKi:  112nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279956(2-Mercaptomethyl-3-o-tolyl-propionic acid | CHEMBL...)
Affinity DataKi:  120nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279961(3-(4-Bromo-phenyl)-2-mercaptomethyl-propionic acid...)
Affinity DataKi:  150nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279963(3-(4-Chloro-phenyl)-2-mercaptomethyl-propionic aci...)
Affinity DataKi:  160nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279953(2-Mercaptomethyl-3-m-tolyl-propionic acid | CHEMBL...)
Affinity DataKi:  170nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279949(2-Mercaptomethyl-3-naphthalen-2-yl-propionic acid ...)
Affinity DataKi:  200nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279945(3-(3,4-Difluoro-phenyl)-2-mercaptomethyl-propionic...)
Affinity DataKi:  250nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279950(3-(2,3-Dimethyl-phenyl)-2-mercaptomethyl-propionic...)
Affinity DataKi:  350nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279957(2-Mercaptomethyl-3-naphthalen-1-yl-propionic acid ...)
Affinity DataKi:  480nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279952(3-(3,4-Dimethyl-phenyl)-2-mercaptomethyl-propionic...)
Affinity DataKi:  492nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279946(2-Mercaptomethyl-3-(3,4,5-trifluoro-phenyl)-propio...)
Affinity DataKi:  590nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279962(2-Mercaptomethyl-3-phenyl-pentanoic acid | CHEMBL1...)
Affinity DataKi:  1.50E+3nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279951(2-Mercaptomethyl-3-pentafluorophenyl-propionic aci...)
Affinity DataKi:  2.30E+3nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50109602(3-Cyclohexyl-2-mercaptomethyl-propionic acid | CHE...)
Affinity DataKi:  2.35E+3nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279959(3-(4-Isopropyl-phenyl)-2-mercaptomethyl-propionic ...)
Affinity DataKi:  4.50E+3nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarboxypeptidase A1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50279948(3-(4-tert-Butyl-phenyl)-2-mercaptomethyl-propionic...)
Affinity DataKi:  7.70E+3nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099832(CHEMBL3319587)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099830(CHEMBL3319585)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099659(CHEMBL3319478)
Affinity DataIC50:  2nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099831(CHEMBL3319586)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50524277(CHEMBL4451741)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of 20S proteasome beta5 subunit in human RPMI8226 cell lysate using Suc-LLVY-AMC as substrate pretreated for 1 hr followed by substrate ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099663(CHEMBL3319482)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50277889(CARFILZOMIB | CHEMBL451887)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of 20S proteasome beta5 subunit in human RPMI8226 cell lysate using Suc-LLVY-AMC as substrate pretreated for 1 hr followed by substrate ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099829(CHEMBL3319584)
Affinity DataIC50:  3nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099685(CHEMBL3319578)
Affinity DataIC50:  3nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099660(CHEMBL3319479)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099833(CHEMBL3319588)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099683(CHEMBL3319484)
Affinity DataIC50:  5nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099687(CHEMBL3319580)
Affinity DataIC50:  5nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099662(CHEMBL3319481)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50277889(CARFILZOMIB | CHEMBL451887)
Affinity DataIC50:  7nMAssay Description:Inhibition of human 20S proteasome chymotrypsin-like activity in human RPMI-8226 cells using Suc-LLVY-AMC as fluorogenic substrate incubated for 3 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50524278(CHEMBL4449204)
Affinity DataIC50:  8nMAssay Description:Inhibition of 20S proteasome beta5 subunit in human RPMI8226 cell lysate using Suc-LLVY-AMC as substrate pretreated for 1 hr followed by substrate ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099664(CHEMBL3319483)
Affinity DataIC50:  8.30nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099686(CHEMBL3319579)
Affinity DataIC50:  11nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099827(CHEMBL3319582)
Affinity DataIC50:  13nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099828(CHEMBL3319583)
Affinity DataIC50:  14nMAssay Description:Inhibition of proteasome subunit beta-5i in human Raji cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50:  18nMAssay Description:Inhibition of proteasome subunit beta-5i in human RPMI8226 cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-9(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099945(CHEMBL3319599)
Affinity DataIC50:  22nMAssay Description:Inhibition of proteasome subunit beta-1i in human Raji cells using BODIPY- epoxomicin by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-9(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50538158(CHEMBL4632784)
Affinity DataIC50:  22nMAssay Description:Inhibition of LMP2 in human 20S immunoproteasome using Ac-PAL-AMC as substrate after 1 hr by fluorescence based microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50099663(CHEMBL3319482)
Affinity DataIC50:  25nMAssay Description:Inhibition of proteasome subunit beta-5i in human RPMI8226 cells using BODIPY-NC005 by fluorescent densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-9(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50573691(CHEMBL4845896)
Affinity DataIC50:  28nMAssay Description:Inhibition of human 20S proteasome LMP2 activity in human RPMI-8226 cells using Ac-PAL-AMC as fluorogenic substrate incubated for 72 hrs by fluoresce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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