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Found 290 with Last Name = 'koltun' and Initial = 'do'
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257967(CHEMBL494748 | N-(2-(7-(4-chloro-3-(trifluoromethy...)
Affinity DataIC50:  0.0500nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257967(CHEMBL494748 | N-(2-(7-(4-chloro-3-(trifluoromethy...)
Affinity DataIC50:  0.0500nMAssay Description:Inhibition of stearoyl-CoA delta9 desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50298907(CHEMBL572876 | N-(2-(6-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of stearoyl-CoA delta9 desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50257967(CHEMBL494748 | N-(2-(7-(4-chloro-3-(trifluoromethy...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of stearoyl-CoA delta9 desaturase in rat microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50298907(CHEMBL572876 | N-(2-(6-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of stearoyl-CoA delta9 desaturase in rat microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50298904(2-hydroxy-N-(2-(2-oxo-3-(trifluoromethyl)-7-(3-(tr...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of stearoyl-CoA delta9 desaturase in rat microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50298904(2-hydroxy-N-(2-(2-oxo-3-(trifluoromethyl)-7-(3-(tr...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of stearoyl-CoA delta9 desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257758(3-(2-(4-methoxyphenyl)-3-oxo-6-(3-(trifluoromethyl...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257968(CHEMBL494359 | N-(2-(7-(4-fluoro-3-methylbenzylami...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257922(CHEMBL494544 | N-(2-(3-(4-ethylphenyl)-2-oxo-7-(3-...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257920(CHEMBL493961 | N-(2-(3-(4-methoxyphenyl)-2-oxo-7-(...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258152(3-(6-(4-methoxyphenyl)-7-oxo-2-(3-(trifluoromethyl...)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50298898(2-hydroxy-N-(2-(3-methyl-2-oxo-7-(3-(trifluorometh...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of stearoyl-CoA delta9 desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258016(CHEMBL522160 | N-(2-(3-(4-methoxyphenyl)-2-oxo-7-(...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257919(CHEMBL493960 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of stearoyl-CoA delta9 desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257919(CHEMBL493960 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258196(3-(7-oxo-6-p-tolyl-2-(3-(trifluoromethyl)benzylami...)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50298909(CHEMBL573830 | N-(2-(6-(3,4-dichlorobenzylamino)-2...)
Affinity DataIC50:  12nMAssay Description:Inhibition of stearoyl-CoA delta9 desaturase in rat microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257809(CHEMBL495170 | N-(2-(6-(3-chloro-4-fluorobenzylami...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257965(CHEMBL494552 | N-(2-(3-(4-methoxyphenyl)-7-(3-meth...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257921(CHEMBL494543 | N-(2-(2-oxo-3-(pyridin-3-yl)-7-(3-(...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50298903(1-(2-(3-methyl-2-oxo-7-(3-(trifluoromethyl)benzyla...)
Affinity DataIC50:  15nMAssay Description:Inhibition of stearoyl-CoA delta9 desaturase in rat microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257808(CHEMBL495001 | N-(2-(6-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257553(CHEMBL523668 | N-(2-(6-(4-fluoro-3-(trifluoromethy...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257757(3-(6-(3,4-dichlorobenzylamino)-2-(4-methoxyphenyl)...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257861(CHEMBL495359 | N-(2-(7-(3,4-dichlorobenzylamino)-2...)
Affinity DataIC50:  21nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257758(3-(2-(4-methoxyphenyl)-3-oxo-6-(3-(trifluoromethyl...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257967(CHEMBL494748 | N-(2-(7-(4-chloro-3-(trifluoromethy...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257919(CHEMBL493960 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257860(CHEMBL495194 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257808(CHEMBL495001 | N-(2-(6-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257758(3-(2-(4-methoxyphenyl)-3-oxo-6-(3-(trifluoromethyl...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257757(3-(6-(3,4-dichlorobenzylamino)-2-(4-methoxyphenyl)...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258197(CHEMBL495191 | N-(2-(6-(3,4-dichlorobenzylamino)-2...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258014(CHEMBL494750 | N-(2-(2-(3,4-dichlorobenzylamino)-6...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257967(CHEMBL494748 | N-(2-(7-(4-chloro-3-(trifluoromethy...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257919(CHEMBL493960 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257860(CHEMBL495194 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257808(CHEMBL495001 | N-(2-(6-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257757(3-(6-(3,4-dichlorobenzylamino)-2-(4-methoxyphenyl)...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258197(CHEMBL495191 | N-(2-(6-(3,4-dichlorobenzylamino)-2...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258014(CHEMBL494750 | N-(2-(2-(3,4-dichlorobenzylamino)-6...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257920(CHEMBL493961 | N-(2-(3-(4-methoxyphenyl)-2-oxo-7-(...)
Affinity DataIC50:  33nMAssay Description:Inhibition of stearoyl-CoA delta9 desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257860(CHEMBL495194 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50:  34nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258154(3-(2-(3,4-dichlorobenzylamino)-7-oxo-6-(pyridin-3-...)
Affinity DataIC50:  36nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50298898(2-hydroxy-N-(2-(3-methyl-2-oxo-7-(3-(trifluorometh...)
Affinity DataIC50:  38nMAssay Description:Inhibition of stearoyl-CoA delta9 desaturase in rat microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257862(CHEMBL522883 | N-(2-(7-(3,4-dichlorobenzylamino)-2...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258240(CHEMBL494031 | N-(2-(6-(3-chloro-4-fluorobenzylami...)
Affinity DataIC50:  47nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258241(CHEMBL494032 | N-(2-(2-(4-methoxyphenyl)-3-oxo-6-(...)
Affinity DataIC50:  47nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50259220(CHEMBL467091 | N-(3-(3,4-dichlorobenzyl)-4-oxo-3,4...)
Affinity DataIC50:  49nMAssay Description:Inhibition of delta(9)-desaturase from human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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