Affinity DataKi: 0.190nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.195nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nM ΔG°: -55.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 0.220nM ΔG°: -55.1kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.370nM ΔG°: -53.8kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from human H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from rat H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 0.501nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.560nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.603nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
Affinity DataKi: 0.692nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.720nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from rat H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.776nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.776nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.851nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Binding affinity for rat histamine H3 receptor on rat cortical cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Antagonist activity at rat histamine H3 receptor expressed in HEK239 cells assessed as inhibition of RAMH-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from rat H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.930nMAssay Description:Displacement of [3H]-N-alpha methyl histamine from rat H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair