Affinity DataKi: 0.230nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 13.4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.62E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.23E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.53E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.84E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 5.06E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 550nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 1.85E+4nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Agonist activity at PPARalpha assessed as receptor transactivation by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Agonist activity at PPARalpha assessed as receptor transactivation by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 1.23E+4nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 2.80E+4nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 1.11E+4nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 60nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 75nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 195nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 1.11E+4nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Mississippi
Curated by ChEMBL
University Of Mississippi
Curated by ChEMBL
Affinity DataEC50: 39nMAssay Description:Transactivation of PPARgamma in CV1 cellsMore data for this Ligand-Target Pair