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Found 84 with Last Name = 'largis' and Initial = 'ee'
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataIC50:  5.30nMAssay Description:Compound was evaluated in vitro for beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50002132((4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethyl...)
Affinity DataIC50:  30nMAssay Description:Compound was evaluated for its binding affinity towards Beta-2 adrenergic receptor in rat soleus membrane by displacing (-)-isoproterenol (50 microM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50002132((4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethyl...)
Affinity DataIC50:  59nMAssay Description:Compound was evaluated for its binding affinity towards Beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227933(CHEMBL77761)
Affinity DataIC50:  140nMAssay Description:In vitro inhibitory concentration against Muscarinic acetylcholine receptor derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50022279(3-(2,4-Difluoro-phenyl)-1-[4-(2,2-dimethyl-propyl)...)
Affinity DataIC50:  140nMAssay Description:Inhibition of smooth muscle cell ACAT activity for cells stimulated by cationized LDL.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50002133((+/-)-2-(4-((R)-2-((R)-2-(3-chlorophenyl)-2-hydrox...)
Affinity DataIC50:  190nMAssay Description:Compound was evaluated in vitro for beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227908(CHEMBL77988)
Affinity DataIC50:  311nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227935(CHEMBL75708)
Affinity DataIC50:  330nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227908(CHEMBL77988)
Affinity DataIC50:  406nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227910(CHEMBL305937)
Affinity DataIC50:  431nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227918(CHEMBL75224)
Affinity DataIC50:  446nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227912(CHEMBL75204)
Affinity DataIC50:  484nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50002132((4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethyl...)
Affinity DataIC50:  500nMAssay Description:Compound was evaluated in vitro for beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataIC50:  600nMAssay Description:Compound was evaluated for its binding affinity towards beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227931(CHEMBL76938)
Affinity DataIC50:  629nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227921(CHEMBL75709)
Affinity DataIC50:  721nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50022279(3-(2,4-Difluoro-phenyl)-1-[4-(2,2-dimethyl-propyl)...)
Affinity DataIC50:  740nMAssay Description:Compound was evaluated for the effect on Cholesterol O-Acyltransferase (ACAT) in Liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50022279(3-(2,4-Difluoro-phenyl)-1-[4-(2,2-dimethyl-propyl)...)
Affinity DataIC50:  810nMAssay Description:Compound was evaluated for the effect on Cholesterol O-Acyltransferase (ACAT) in intestinal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227943(CHEMBL76935)
Affinity DataIC50:  952nMAssay Description:In vitro inhibitory concentration against ACAT derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227909(CHEMBL307505)
Affinity DataIC50:  976nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Canis familiaris)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataIC50:  1.00E+3nMAssay Description:Compound was evaluated for its binding affinity towards beta-2 adrenergic receptor in rat soleus membrane by displacing(-)-isoproterenol (50 microM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227918(CHEMBL75224)
Affinity DataIC50:  1.08E+3nMAssay Description:In vitro inhibitory concentration against ACAT derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50022279(3-(2,4-Difluoro-phenyl)-1-[4-(2,2-dimethyl-propyl)...)
Affinity DataIC50:  1.09E+3nMAssay Description:Compound was evaluated for the effect on Cholesterol O-Acyltransferase (ACAT) in Aorta (homogenate Low-density lipoproteins (LDL)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50002133((+/-)-2-(4-((R)-2-((R)-2-(3-chlorophenyl)-2-hydrox...)
Affinity DataIC50:  1.30E+3nMAssay Description:Compound was evaluated for its binding affinity towards Beta-2 adrenergic receptor in rat soleus membrane by displacing (-)-isoproterenol (50 microM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227936(CHEMBL73918)
Affinity DataIC50:  1.31E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227936(CHEMBL73918)
Affinity DataIC50:  1.41E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227907(CHEMBL441803)
Affinity DataIC50:  1.44E+3nMAssay Description:In vitro inhibitory concentration against ACAT derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227902(CHEMBL76706)
Affinity DataIC50:  1.71E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227915(CHEMBL421876)
Affinity DataIC50:  1.83E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227933(CHEMBL77761)
Affinity DataIC50:  2.24E+3nMAssay Description:In vitro inhibitory concentration against Muscarinic acetylcholine receptor derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227909(CHEMBL307505)
Affinity DataIC50:  2.62E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227932(CHEMBL77164)
Affinity DataIC50:  2.86E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227937(CHEMBL76258)
Affinity DataIC50:  3.01E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227948(CHEMBL75596)
Affinity DataIC50:  3.18E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227944(CHEMBL77942)
Affinity DataIC50:  3.28E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50002133((+/-)-2-(4-((R)-2-((R)-2-(3-chlorophenyl)-2-hydrox...)
Affinity DataIC50:  3.30E+3nMAssay Description:Compound was evaluated for its binding affinity towards Beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227929(CHEMBL419639)
Affinity DataIC50:  3.54E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227934(CHEMBL75371)
Affinity DataIC50:  3.62E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227906(CHEMBL74091)
Affinity DataIC50:  3.62E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227902(CHEMBL76706)
Affinity DataIC50:  3.77E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227917(CHEMBL77694)
Affinity DataIC50:  3.89E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227925(CHEMBL75331)
Affinity DataIC50:  4.04E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227927(CHEMBL442178)
Affinity DataIC50:  4.41E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227910(CHEMBL305937)
Affinity DataIC50:  4.53E+3nMAssay Description:In vitro inhibitory concentration against Acyl coenzyme A:cholesterol acyltransferase derived from smooth muscle cells from thoracic aorta of monkeysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227923(CHEMBL305913)
Affinity DataIC50:  4.59E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227915(CHEMBL421876)
Affinity DataIC50:  4.83E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227924(CHEMBL307709)
Affinity DataIC50:  4.95E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227928(CHEMBL75354)
Affinity DataIC50:  5.64E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50227930(CHEMBL77943)
Affinity DataIC50:  5.81E+3nMAssay Description:In vitro inhibitory concentration against acyl coenzyme A:cholesterol acyltransferase derived from rat adrenalsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50022279(3-(2,4-Difluoro-phenyl)-1-[4-(2,2-dimethyl-propyl)...)
Affinity DataIC50:  6.06E+3nMAssay Description:Inhibition of smooth muscle cell ACAT activity for cells stimulated by native LDL.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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