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Found 76 with Last Name = 'larsen' and Initial = 'y'
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  390nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2A expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159745(CHEMBL3786901)
Affinity DataKi:  434nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA1 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159745(CHEMBL3786901)
Affinity DataKi:  1.53E+3nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA3 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159745(CHEMBL3786901)
Affinity DataKi:  2.75E+3nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA4 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  2.80E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2B expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159750(CHEMBL3786611)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA1 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  4.70E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2A expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159748(CHEMBL3785581)
Affinity DataKi:  5.29E+3nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA1 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  5.90E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2C expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159745(CHEMBL3786901)
Affinity DataKi:  8.15E+3nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA2 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 3(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159746(CHEMBL3785285)
Affinity DataKi:  8.47E+3nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA3 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  1.00E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2B expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159746(CHEMBL3785285)
Affinity DataKi:  1.08E+4nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA1 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246919(CHEMBL4099104)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246919(CHEMBL4099104)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159750(CHEMBL3786611)
Affinity DataKi:  1.60E+4nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA3 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159752(CHEMBL3786824)
Affinity DataKi:  1.91E+4nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA3 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2D(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  2.10E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2D expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor 3(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159748(CHEMBL3785581)
Affinity DataKi:  2.23E+4nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA3 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  2.40E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2C expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2D(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  4.10E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2D expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159750(CHEMBL3786611)
Affinity DataKi:  5.50E+4nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA2 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159752(CHEMBL3786824)
Affinity DataKi:  5.56E+4nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA4 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159746(CHEMBL3785285)
Affinity DataKi:  8.44E+4nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA2 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159748(CHEMBL3785581)
Affinity DataKi:  8.45E+4nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA2 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159748(CHEMBL3785581)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from recombinant rat GluK2(V,C,R) receptor expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159750(CHEMBL3786611)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from recombinant rat GluK2(V,C,R) receptor expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159752(CHEMBL3786824)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from recombinant rat GluK2(V,C,R) receptor expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50159745(CHEMBL3786901)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from recombinant rat GluK3 receptor expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50159746(CHEMBL3785285)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from recombinant rat GluK3 receptor expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50159748(CHEMBL3785581)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from recombinant rat GluK3 receptor expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50159750(CHEMBL3786611)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from recombinant rat GluK3 receptor expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50159752(CHEMBL3786824)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from recombinant rat GluK3 receptor expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159746(CHEMBL3785285)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from recombinant rat GluK2(V,C,R) receptor expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159745(CHEMBL3786901)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from recombinant rat GluK2(V,C,R) receptor expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159752(CHEMBL3786824)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA2 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159752(CHEMBL3786824)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA1 receptor flop isoform expressed in sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246911(CHEMBL4076785)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246917(CHEMBL4068651)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246915(CHEMBL4060745)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246918(CHEMBL4091369)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50246914(CHEMBL4088958)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50246911(CHEMBL4076785)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246918(CHEMBL4091369)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246916(CHEMBL4102488)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246914(CHEMBL4088958)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246911(CHEMBL4076785)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50246917(CHEMBL4068651)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50246916(CHEMBL4102488)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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