TargetThermolysin(Bacillus thermoproteolyticus)
Pohang University Of Science And Technology
Curated by ChEMBL
Pohang University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 3.40E+4nMpH: 7.2Assay Description:Inhibitory activity against thermolysin using 2-furylacryloyl-Gly-Leu-NH2 as substrate at pH 7.2More data for this Ligand-Target Pair
TargetThermolysin(Bacillus thermoproteolyticus)
Pohang University Of Science And Technology
Curated by ChEMBL
Pohang University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 4.00E+4nMpH: 7.2Assay Description:Inhibitory activity against thermolysin using 2-furylacryloyl-Gly-Leu-NH2 as substrate at pH 7.2More data for this Ligand-Target Pair
TargetThermolysin(Bacillus thermoproteolyticus)
Pohang University Of Science And Technology
Curated by ChEMBL
Pohang University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 5.40E+4nMpH: 7.2Assay Description:Inhibitory activity against thermolysin using 2-furylacryloyl-Gly-Leu-NH2 as substrate at pH 7.2More data for this Ligand-Target Pair
TargetThermolysin(Bacillus thermoproteolyticus)
Pohang University Of Science And Technology
Curated by ChEMBL
Pohang University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 8.20E+4nMpH: 7.2Assay Description:Inhibitory activity against thermolysin using 2-furylacryloyl-Gly-Leu-NH2 as substrate at pH 7.2More data for this Ligand-Target Pair
TargetThermolysin(Bacillus thermoproteolyticus)
Pohang University Of Science And Technology
Curated by ChEMBL
Pohang University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 2.44E+5nMpH: 7.2Assay Description:Inhibitory activity against thermolysin using 2-furylacryloyl-Gly-Leu-NH2 as substrate at pH 7.2More data for this Ligand-Target Pair
TargetThermolysin(Bacillus thermoproteolyticus)
Pohang University Of Science And Technology
Curated by ChEMBL
Pohang University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 3.40E+5nMpH: 7.2Assay Description:Inhibitory activity against thermolysin using 2-furylacryloyl-Gly-Leu-NH2 as substrate at pH 7.2More data for this Ligand-Target Pair
TargetThermolysin(Bacillus thermoproteolyticus)
Pohang University Of Science And Technology
Curated by ChEMBL
Pohang University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 7.74E+5nMpH: 7.2Assay Description:Inhibitory activity against thermolysin using 2-furylacryloyl-Gly-Leu-NH2 as substrate at pH 7.2More data for this Ligand-Target Pair
TargetThermolysin(Bacillus thermoproteolyticus)
Pohang University Of Science And Technology
Curated by ChEMBL
Pohang University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.91E+6nMpH: 7.2Assay Description:Inhibitory activity against thermolysin using 2-furylacryloyl-Gly-Leu-NH2 as substrate at pH 7.2More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of rat Nav1.7 stably expressed in cells with train pulses to -20 mV at 0.1 Hz and holding potential of -90 mV by whole-cell QPatch HT assa...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into GST-ATF2 substrate preincubated for 20 mins before substrate addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human Nav1.7 stably expressed in cells with train pulses to -20 mV at 0.1 Hz and holding potential of -95 mV by whole-cell QPatch HT as...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]-E2 from estrogen receptor-beta (unknown origin) by scintillation counting analysisMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Inhibition of human Nav1.7 stably expressed in cells with train pulses to -20 mV at 0.1 Hz and holding potential of -95 mV by whole-cell QPatch HT as...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]-E2 from estrogen receptor-alpha (unknown origin) by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into GST-ATF2 substrate preincubated for 20 mins before substrate addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Displacement of [3H]-E2 from estrogen receptor-alpha (unknown origin) by scintillation counting analysisMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Inhibition of rat Nav1.7 stably expressed in cells with train pulses to -20 mV at 0.1 Hz and holding potential of -90 mV by whole-cell QPatch HT assa...More data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Displacement of [3H]-E2 from estrogen receptor-beta (unknown origin) by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into GST-ATF2 substrate preincubated for 20 mins before substrate addition measured a...More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of JNK2alpha2More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into GST-ATF2 substrate preincubated for 20 mins before substrate addition measured a...More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into GST-ATF2 substrate preincubated for 20 mins before substrate addition measured a...More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into GST-ATF2 substrate preincubated for 20 mins before substrate addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into GST-ATF2 substrate preincubated for 20 mins before substrate addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into GST-ATF2 substrate preincubated for 20 mins before substrate addition measured a...More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair