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Found 228 with Last Name = 'liclican' and Initial = 'a'
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230294(CHEMBL4071740)
Affinity DataKi:  4nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230211(CHEMBL4063126)
Affinity DataKi:  4.30nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataKi:  6.70nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230212(CHEMBL4084776)
Affinity DataKi:  7nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230213(CHEMBL4092526)
Affinity DataKi:  14nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230210(CHEMBL4090107)
Affinity DataKi:  16nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230209(CHEMBL4100272)
Affinity DataKi:  65nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Selcia

Curated by ChEMBL
LigandPNGBDBM50230293(CHEMBL4082253)
Affinity DataKi:  795nMAssay Description:Inhibition of full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed in Escherichia coli BL21(DE3) using Su...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315949((S)-N-(4-aminobutyl)-N-(2-(1-phenylethylamino)pyri...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306491(2-(6-chloro-5-((2R,5S)-4-(1-(4-fluorophenyl)ethyl)...)
Affinity DataIC50:  6nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306493(2-(5-((2R,5S)-4-benzhydryl-2,5-dimethylpiperazine-...)
Affinity DataIC50:  9nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50266947(2-(6-chloro-5-((2R,5S)-4-(4-fluorobenzyl)-2,5-dime...)
Affinity DataIC50:  9nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
LigandPNGBDBM50374977(CHEMBL270849)
Affinity DataIC50:  9nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375063(CHEMBL255607)
Affinity DataIC50:  10nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50309525(2-(5-(4-(4-fluorobenzyl)piperidine-1-carbonyl)-6-m...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315959(CHEMBL1091614 | N-(4-aminobutyl)-N-(2-(4-hydroxycy...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374956(CHEMBL272978)
Affinity DataIC50:  12nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315931((S)-N-ethyl-3-methyl-N-(2-(1-phenylethylamino)pyri...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375073(CHEMBL402340)
Affinity DataIC50:  13nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315917((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315958(CHEMBL1089655 | N-(4-aminobutyl)-N-(2-(isopropylam...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50309524(2-(6-chloro-5-(4-(4-fluorobenzyl)piperidine-1-carb...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375061(CHEMBL271648)
Affinity DataIC50:  21nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315951(CHEMBL1093834 | N-(2-(isopropylamino)pyrimidin-4-y...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306492(2-(5-((2R,5S)-4-(bis(4-fluorophenyl)methyl)-2,5-di...)
Affinity DataIC50:  24nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315960((S)-N-(4-aminobutyl)-N-(2-(1-methoxypropan-2-ylami...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315938((S)-N-ethyl-2-fluoro-5-methyl-N-(2-(1-phenylethyla...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306494(2-(6-chloro-5-((2R,5S)-4-(2,3-dihydro-1H-inden-1-y...)
Affinity DataIC50:  29nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375062(CHEMBL402533)
Affinity DataIC50:  32nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374982(CHEMBL403446)
Affinity DataIC50:  34nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374982(CHEMBL403446)
Affinity DataIC50:  34nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375072(CHEMBL403337)
Affinity DataIC50:  38nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315937((S)-N-ethyl-4-fluoro-3-methyl-N-(2-(1-phenylethyla...)
Affinity DataIC50:  39nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374954(CHEMBL271045)
Affinity DataIC50:  42nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315922((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)
Affinity DataIC50:  45nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375071(CHEMBL270032)
Affinity DataIC50:  46nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306496(2-(6-chloro-5-((2R,5S)-4-(1-cyano-1-(4-fluoropheny...)
Affinity DataIC50:  47nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306497(2-(6-chloro-5-((2R,5S)-4-(7-chloro-1H-indazol-3-yl...)
Affinity DataIC50:  48nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315943((S)-N-(2-(1-phenylethylamino)pyrimidin-4-yl)-N-(pi...)
Affinity DataIC50:  54nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50309531(2-(5-(4-(4-fluorobenzyl)piperidine-1-carbonyl)-6-m...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315916((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315936((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374963(CHEMBL402428)
Affinity DataIC50:  64nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315934((S)-N,3-diethyl-N-(2-(1-phenylethylamino)pyrimidin...)
Affinity DataIC50:  65nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374965(CHEMBL255617)
Affinity DataIC50:  66nMAssay Description:Inhibition of cloned CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315920((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)
Affinity DataIC50:  71nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315919((S)-N-(3-(methylsulfonyl)propyl)-N-(2-(1-phenyleth...)
Affinity DataIC50:  72nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315933((S)-N-ethyl-2,3-dimethyl-N-(2-(1-phenylethylamino)...)
Affinity DataIC50:  81nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315929((S)-3-chloro-N-ethyl-N-(2-(1-phenylethylamino)pyri...)
Affinity DataIC50:  81nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50315921((S)-N-ethyl-N-(2-(1-phenylethylamino)pyrimidin-4-y...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human p38alpha assessed as gamma-[32P]ATP incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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