TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.0420nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO/HEK293 cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.0680nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.0860nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.0910nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.0940nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Inhibition of [125I]-iodoproxyfan from rat histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:In vitro inhibitory activity against Histamine H3 receptor for K+ evoked depolarization-induced release of [3H]-histamine from synaptosomes of rat ce...More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO/HEK293 cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Histamine H3 receptor antagonist activity in an assay with K+ evoked depolarization-induced release of [3H]-histamine from rat synaptosomes.More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.260nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.260nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Displacement of [125I]Iodoproxyfan from mouse brain cortex histamine H3 receptor after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Histamine H3 receptor antagonist activity in an assay with K+ evoked depolarization-induced release of [3H]-histamine from rat synaptosomes.More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.320nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Displacement of [125I]Iodoproxyfan from mouse brain cortex histamine H3 receptor after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.358nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO/HEK293 cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Histamine H3 receptor antagonist activity in an assay with K+ evoked depolarization-induced release of [3H]-histamine from rat synaptosomes.More data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Histamine H3 receptor antagonist activity in an assay with K+ evoked depolarization-induced release of [3H]-histamine from rat synaptosomes.More data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:In vitro inhibitory activity against Histamine H3 receptor for K+ evoked depolarization-induced release of [3H]-histamine from synaptosomes of rat ce...More data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Histamine H3 receptor antagonist activity in an assay with K+ evoked depolarization-induced release of [3H]-histamine from rat synaptosomes.More data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Effect on histamine H3 receptors in vitro, on synaptosomes of rat cerebral cortex for the release of [3H]histamineMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:In vitro binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:Displacement of [125I]Iodoproxyfan from mouse brain cortex histamine H3 receptor after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.530nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.530nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.560nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.570nMAssay Description:Displacement of [125I]Iodoproxyfan from recombinant human histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Johann Wolfgang Goethe Universit£T
Curated by ChEMBL
Affinity DataKi: 0.580nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair